BG61420B2 - 3-метилов естер 5-етилов естер на 2,6-диметил-4-(2,3- дихлорофенил)-1,4-дихидропиридин-3,5-дикарбоксиловата киселина,притежаващ хипотензивни свойства,метод за неговото получаване и фармацевтични пре парати, които ги съдържат - Google Patents

3-метилов естер 5-етилов естер на 2,6-диметил-4-(2,3- дихлорофенил)-1,4-дихидропиридин-3,5-дикарбоксиловата киселина,притежаващ хипотензивни свойства,метод за неговото получаване и фармацевтични пре парати, които ги съдържат Download PDF

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Publication number
BG61420B2
BG61420B2 BG098595A BG9859594A BG61420B2 BG 61420 B2 BG61420 B2 BG 61420B2 BG 098595 A BG098595 A BG 098595A BG 9859594 A BG9859594 A BG 9859594A BG 61420 B2 BG61420 B2 BG 61420B2
Authority
BG
Bulgaria
Prior art keywords
compound
formula
dimethyl
dihydropyridine
methyl ester
Prior art date
Application number
BG098595A
Other languages
Bulgarian (bg)
English (en)
Inventor
Peter Berntsson
Stig Ake Carlsson
Jan Gaarden
Bengt Ljung
Original Assignee
Aktiebolaget Haessle
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20335348&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG61420(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aktiebolaget Haessle filed Critical Aktiebolaget Haessle
Publication of BG61420B2 publication Critical patent/BG61420B2/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG098595A 1978-06-30 1994-02-25 3-метилов естер 5-етилов естер на 2,6-диметил-4-(2,3- дихлорофенил)-1,4-дихидропиридин-3,5-дикарбоксиловата киселина,притежаващ хипотензивни свойства,метод за неговото получаване и фармацевтични пре парати, които ги съдържат BG61420B2 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE7807404A SE429652B (sv) 1978-06-30 1978-06-30 2.6-dimetyl-4-(2.3-diklorfenyl)-1.4-dihydropyridin-3.5-dikarboxylsyra-3-metylester-5-etylester

Publications (1)

Publication Number Publication Date
BG61420B2 true BG61420B2 (bg) 1997-07-31

Family

ID=20335348

Family Applications (1)

Application Number Title Priority Date Filing Date
BG098595A BG61420B2 (bg) 1978-06-30 1994-02-25 3-метилов естер 5-етилов естер на 2,6-диметил-4-(2,3- дихлорофенил)-1,4-дихидропиридин-3,5-дикарбоксиловата киселина,притежаващ хипотензивни свойства,метод за неговото получаване и фармацевтични пре парати, които ги съдържат

Country Status (24)

Country Link
US (1) US4264611A (instruction)
EP (1) EP0007293B1 (instruction)
JP (1) JPS559083A (instruction)
AT (1) ATE1237T1 (instruction)
AU (1) AU529116B2 (instruction)
BG (1) BG61420B2 (instruction)
CA (1) CA1117530A (instruction)
CS (1) CS241021B2 (instruction)
CY (1) CY1299A (instruction)
DD (1) DD144667A5 (instruction)
DE (1) DE2963150D1 (instruction)
DK (1) DK148978C (instruction)
FI (1) FI70573C (instruction)
HK (1) HK60585A (instruction)
HU (1) HU178568B (instruction)
IE (1) IE48650B1 (instruction)
LU (2) LU88666I2 (instruction)
NL (2) NL930054I2 (instruction)
NO (3) NO151965C (instruction)
NZ (1) NZ190809A (instruction)
SE (1) SE429652B (instruction)
SG (1) SG26085G (instruction)
SU (2) SU856380A3 (instruction)
ZA (1) ZA792804B (instruction)

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DE4342196A1 (de) * 1993-12-10 1995-06-14 Bayer Ag Neue 4-Phenyl-substituierte 1,4-Dihydropyridine
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RU2570752C2 (ru) 2011-08-26 2015-12-10 Вокхардт Лимитед Способы лечения сердечно-сосудистых нарушений
CN105143203A (zh) 2013-04-17 2015-12-09 辉瑞大药厂 用于治疗心血管疾病的n-哌啶-3-基苯甲酰胺衍生物
CN104177286A (zh) * 2014-08-11 2014-12-03 广东东阳光药业有限公司 一种地平类药物的制备方法
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Also Published As

Publication number Publication date
LU88306I2 (fr) 1994-05-04
IE791217L (en) 1979-12-30
ZA792804B (en) 1980-06-25
NO1994026I1 (no) 1994-12-21
CY1299A (en) 1985-10-18
NZ190809A (en) 1982-03-09
NO1996006I1 (no) 1996-06-24
DE2963150D1 (en) 1982-08-12
ATE1237T1 (de) 1982-07-15
SG26085G (en) 1986-01-24
SU915799A3 (en) 1982-03-23
DD144667A5 (de) 1980-10-29
AU4831679A (en) 1980-02-07
EP0007293B1 (en) 1982-06-23
SE7807404L (sv) 1979-12-31
AU529116B2 (en) 1983-05-26
HK60585A (en) 1985-08-23
JPS559083A (en) 1980-01-22
HU178568B (en) 1982-05-28
NO151965B (no) 1985-04-01
NO792112L (no) 1980-01-03
CA1117530A (en) 1982-02-02
IE48650B1 (en) 1985-04-03
NL930054I1 (nl) 1993-09-01
NL940012I1 (nl) 1994-08-01
FI792058A7 (fi) 1979-12-31
SU856380A3 (ru) 1981-08-15
EP0007293A1 (en) 1980-01-23
DK148978B (da) 1985-12-09
CS241021B2 (en) 1986-03-13
US4264611A (en) 1981-04-28
US4264611B1 (instruction) 1984-07-17
LU88666I2 (fr) 1996-02-01
SE429652B (sv) 1983-09-19
NO151965C (no) 1985-07-10
FI70573C (fi) 1986-09-24
DK275079A (da) 1979-12-31
NL930054I2 (nl) 1994-02-16
FI70573B (fi) 1986-06-06
DK148978C (da) 1986-08-18
JPS6121550B2 (instruction) 1986-05-27

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