BE762135A - Nouvelles 4-morpholino-thieno-(3,2-d)pyrimidines et procede pour les fabriquer - Google Patents
Nouvelles 4-morpholino-thieno-(3,2-d)pyrimidines et procede pour les fabriquerInfo
- Publication number
- BE762135A BE762135A BE762135A BE762135A BE762135A BE 762135 A BE762135 A BE 762135A BE 762135 A BE762135 A BE 762135A BE 762135 A BE762135 A BE 762135A BE 762135 A BE762135 A BE 762135A
- Authority
- BE
- Belgium
- Prior art keywords
- thieno
- pyrimidines
- morpholino
- news
- manufacturing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19702003714 DE2003714C (de) | 1970-01-28 | 2 Piperazino 4 morpholino thieno eckige Klammer auf 3,2 d eckige Klammer zu pyrimidin und dessen Saureadditions salze | |
DE19702058086 DE2058086A1 (de) | 1970-11-26 | 1970-11-26 | Neue 4-Morpholino-thieno[3,2-d]pyrimidine,deren Salze und Verfahren zur Herstellung |
DE19702058085 DE2058085A1 (de) | 1970-11-26 | 1970-11-26 | Neues Verfahren zur Herstellung von 4-Morpholino-thieno[3,2-d]pyrimidinen |
Publications (1)
Publication Number | Publication Date |
---|---|
BE762135A true BE762135A (fr) | 1971-07-27 |
Family
ID=27182372
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE762135A BE762135A (fr) | 1970-01-28 | 1971-01-27 | Nouvelles 4-morpholino-thieno-(3,2-d)pyrimidines et procede pour les fabriquer |
Country Status (9)
Country | Link |
---|---|
US (1) | US3763156A (de) |
AU (1) | AU2468871A (de) |
BE (1) | BE762135A (de) |
ES (2) | ES387553A1 (de) |
FR (1) | FR2081464B1 (de) |
GB (1) | GB1309182A (de) |
IL (1) | IL36079A0 (de) |
NL (1) | NL7101043A (de) |
NO (1) | NO129205B (de) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1570494A (en) * | 1975-11-28 | 1980-07-02 | Ici Ltd | Thienopyrimidine derivatives and their use as pesticides |
US5280026A (en) * | 1989-05-30 | 1994-01-18 | Smithkline Beecham Intercredit B.V. | Thienopyrimidines |
GB8912335D0 (en) * | 1989-05-30 | 1989-07-12 | Smithkline Beckman Intercredit | Compounds |
US5098902A (en) * | 1991-03-18 | 1992-03-24 | Warner-Lambert Company | Method of treating neurodegenerative diseases |
US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
US6608053B2 (en) * | 2000-04-27 | 2003-08-19 | Yamanouchi Pharmaceutical Co., Ltd. | Fused heteroaryl derivatives |
GB0423653D0 (en) * | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
RS51163B (sr) * | 2006-04-19 | 2010-10-31 | Boehringer Ingelheim International Gmbh. | Dihidrotienopirimidin za lečenje zapaljenskih bolesti |
EP1847543A1 (de) | 2006-04-19 | 2007-10-24 | Boehringer Ingelheim Pharma GmbH & Co. KG | Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen |
NZ572812A (en) * | 2006-04-26 | 2010-09-30 | Hoffmann La Roche | THIENO [3, 2-D] PYRIMIDINE Indazole DERIVATIVE USEFUL AS PI3K INHIBITOR |
ATE532788T1 (de) * | 2006-04-26 | 2011-11-15 | Hoffmann La Roche | Pharmazeutische verbindungen |
CL2007001166A1 (es) | 2006-04-26 | 2008-01-25 | Piramed Ltd | Compuestos derivados de pirimidina condensada, inhibidores de pi3-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicion farmaceutica |
ES2544082T3 (es) * | 2006-12-07 | 2015-08-27 | F. Hoffmann-La Roche Ag | Compuestos inhibidores de fosfoinosítido 3-quinasa y métodos de uso |
EP2114950B1 (de) * | 2006-12-07 | 2016-03-09 | Genentech, Inc. | Phosphoinositid-3-kinaseinhibitorverbindungen und anwendungsverfahren |
EP2207781B1 (de) | 2007-09-24 | 2012-11-28 | Genentech, Inc. | Thiazolopyrimidinverbindungen als p13k-inhibitoren und anwendungsverfahren |
EP2215093B1 (de) | 2007-10-19 | 2011-12-14 | Boehringer Ingelheim International GmbH | Neue piperazino-dihydrothienopyrimidin-derivate |
MX2010004026A (es) * | 2007-10-19 | 2010-04-30 | Boehringer Ingelheim Int | Piperidino-dihidrotienopirimidinas sustituidas. |
EP2205609B1 (de) | 2007-10-19 | 2017-03-29 | Boehringer Ingelheim International GmbH | Heterocyclus-substituierte piperazino-dihydrothienopyrimidine |
EP2214675B1 (de) | 2007-10-25 | 2013-11-20 | Genentech, Inc. | Verfahren zur herstellung von thienopyrimidin-verbindungen |
GB0721095D0 (en) * | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
CN102369011A (zh) | 2009-03-12 | 2012-03-07 | 健泰科生物技术公司 | 用于治疗造血恶性肿瘤的磷酸肌醇3-激酶抑制剂化合物与化学治疗剂的组合 |
JP5781066B2 (ja) | 2009-05-27 | 2015-09-16 | ジェネンテック, インコーポレイテッド | p110δに対して選択的な二環式ピリミジンPI3K阻害剤化合物及び使用方法 |
US8158625B2 (en) * | 2009-05-27 | 2012-04-17 | Genentech, Inc. | Bicyclic indole-pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use |
MX345155B (es) * | 2009-10-12 | 2017-01-18 | F Hoffmann-La Roche Ag * | Combinaciones de un inhibidor de pi3k y un inhibidor de mek. |
EP2558864A1 (de) | 2010-04-16 | 2013-02-20 | Genentech, Inc. | Fox03a als prädiktiver biomarker zur hemmung des pi3k/akt-kinasesignalweges |
US20140004209A1 (en) | 2010-12-22 | 2014-01-02 | Genentech, Inc. | Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms |
US9802954B2 (en) | 2011-08-24 | 2017-10-31 | Boehringer Ingelheim International Gmbh | Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma |
US20130059866A1 (en) | 2011-08-24 | 2013-03-07 | Boehringer Ingelheim International Gmbh | Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma |
CN105247072B (zh) | 2013-02-25 | 2019-10-15 | 基因泰克公司 | 检测和治疗抗药性akt突变体的方法和组合物 |
US11098056B2 (en) * | 2018-10-01 | 2021-08-24 | Genzyme Corporation | UDP glycosyltransferase inhibitors and methods of use |
GB202014736D0 (en) * | 2020-09-18 | 2020-11-04 | Imperial College Innovations Ltd | Novel compounds and their use in therapy |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1470356A1 (de) * | 1964-01-15 | 1970-04-30 | Thomae Gmbh Dr K | Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
-
1971
- 1971-01-22 US US00108988A patent/US3763156A/en not_active Expired - Lifetime
- 1971-01-23 ES ES387553A patent/ES387553A1/es not_active Expired
- 1971-01-23 ES ES387554A patent/ES387554A1/es not_active Expired
- 1971-01-26 AU AU24688/71A patent/AU2468871A/en not_active Expired
- 1971-01-27 NL NL7101043A patent/NL7101043A/xx unknown
- 1971-01-27 NO NO00283/71A patent/NO129205B/no unknown
- 1971-01-27 BE BE762135A patent/BE762135A/xx unknown
- 1971-01-27 IL IL36079A patent/IL36079A0/xx unknown
- 1971-01-28 FR FR7102796A patent/FR2081464B1/fr not_active Expired
- 1971-04-19 GB GB2046471A patent/GB1309182A/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
IL36079A0 (en) | 1971-03-24 |
AU2468871A (en) | 1972-07-27 |
ES387554A1 (es) | 1974-01-16 |
ES387553A1 (es) | 1974-01-16 |
NO129205B (de) | 1974-03-11 |
FR2081464B1 (de) | 1975-04-18 |
GB1309182A (en) | 1973-03-07 |
FR2081464A1 (de) | 1971-12-03 |
NL7101043A (de) | 1971-07-30 |
US3763156A (en) | 1973-10-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BE762135A (fr) | Nouvelles 4-morpholino-thieno-(3,2-d)pyrimidines et procede pour les fabriquer | |
BE779203A (fr) | 2-hydrocarbyldithio-5-mercapto-1, 3, 4, -thiadiazoles et procede pour les preparer, | |
CH550476A (fr) | Element dielectrique et procede pour le fabriquer. | |
BE783044A (fr) | Nouvelles thieno(3,2-d) pyrimidines | |
BE759493A (fr) | Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer | |
BE768898A (fr) | Procede d'ajustement de capacites | |
BE776958R (fr) | Tetra-oxo-1,2-dipiperazino-alcanes et procede pour leur | |
BE761232A (fr) | Electrodes pour elements au ni-cd et procede de leur fabrication | |
BE776969A (fr) | Nouvelles phenoxyalcoylamines, leur procede de preparation et leurs applications | |
BE761321A (fr) | Nouvelles amines et procede pour leur preparation | |
BE768403A (fr) | Nouvelles aminophenylamidines vermifuges et procede pour leur obtentio | |
IT953448B (it) | Metodo per produrre seleniuri di arsenico e selenio drogato con arsenico | |
OA03675A (fr) | Eléments de fondation et/ou de soutènement et procédé pour les fabriquer. | |
BE808599A (fr) | Nouvelles pyrazolodiazepines et procede pour les preparer | |
BE746576A (fr) | Ethers de 4.20.22-bufatrienolidrhamnoside et procede pour les preparer | |
BE748770A (fr) | Nouveaux ethers basiques et procede pour les | |
BE794532A (fr) | Nouvelles 3-hydroxymethyl-5-benzylidene-azolidinones et procede pour les fabriquer | |
CH550152A (fr) | Procede de preparation de nouvelles iodomethylsulfones. | |
BE752984A (fr) | Procede de fabrication de la tetrachloropyrimidine | |
BE755689A (fr) | Procede de fabrication de nouvelles 7 beta-alkyl-19- nortestosterones | |
BE758621A (fr) | Nouvelles amidines et leur procede de preparation | |
BE753901A (fr) | Nouvelles benzamidines et procede pour leur preparation | |
BE777238A (fr) | Dioxypiperidines substituees et procede pour les | |
BE800564A (fr) | Nouvelles 3,6-bis-(aminoacylamino)-acridines et procede pour les fabriquer | |
BE750725A (fr) | Nouvelles 2-alcoyloxymethyl-3-chloro-1, 2,4-thiaimidazol-5-oneset procede pour les preparer |