AU6736596A - Prodrugs of 4-{3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl} -4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists - Google Patents

Prodrugs of 4-{3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl} -4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists

Info

Publication number
AU6736596A
AU6736596A AU67365/96A AU6736596A AU6736596A AU 6736596 A AU6736596 A AU 6736596A AU 67365/96 A AU67365/96 A AU 67365/96A AU 6736596 A AU6736596 A AU 6736596A AU 6736596 A AU6736596 A AU 6736596A
Authority
AU
Australia
Prior art keywords
dimethylaminocyclobutyl
oxazolidin
indol
prodrugs
trans
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU67365/96A
Inventor
Robert John Blade
David Lawrence Selwood
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of AU6736596A publication Critical patent/AU6736596A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU67365/96A 1995-07-26 1996-07-24 Prodrugs of 4-{3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl} -4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists Abandoned AU6736596A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9515305.2A GB9515305D0 (en) 1995-07-26 1995-07-26 Therapeutic heterocyclic compounds
GB9515305 1995-07-26
PCT/EP1996/003251 WO1997005133A1 (en) 1995-07-26 1996-07-24 Prodrugs of 4-[3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl]-4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists

Publications (1)

Publication Number Publication Date
AU6736596A true AU6736596A (en) 1997-02-26

Family

ID=10778267

Family Applications (1)

Application Number Title Priority Date Filing Date
AU67365/96A Abandoned AU6736596A (en) 1995-07-26 1996-07-24 Prodrugs of 4-{3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl} -4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists

Country Status (3)

Country Link
AU (1) AU6736596A (en)
GB (1) GB9515305D0 (en)
WO (1) WO1997005133A1 (en)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8601959D0 (en) * 1986-01-28 1986-03-05 Glaxo Group Ltd Indole derivatives
EP0486666B1 (en) * 1990-06-07 1997-08-13 Zeneca Limited Therapeutic heterocyclic compounds
WO1994002477A1 (en) * 1992-07-24 1994-02-03 Merck Sharp & Dohme Limited Imidazole, triazole and tetrazole derivatives
GB9401436D0 (en) * 1994-01-26 1994-03-23 Wellcome Found Therapeutic heterocyclic compounds
JP3262800B2 (en) * 1994-06-01 2002-03-04 ゼネカ・リミテッド Therapeutic heterocyclic compounds

Also Published As

Publication number Publication date
GB9515305D0 (en) 1995-09-20
WO1997005133A1 (en) 1997-02-13

Similar Documents

Publication Publication Date Title
AU654119B2 (en) Isoxazolines, method of preparation thereof, and their use as plant-protection agents
HUP9901629A3 (en) Use of r(+)-enantiomer of n-propargyl-1-aminoindan, salts, and compositions thereof
AU2183900A (en) Ep4 receptor agonists for treatment of dry eye
AU7106096A (en) Catalyst composition and methods for using and preparing same
AU4422293A (en) Substituted 2-amidotetralins as melatonin agonists and antagonists
AU7042396A (en) Maintaining the composition of transferred data during handover
AU4520697A (en) Use of substituted benzazoles as UV absorbers, new benzazoles and processes for their preparation
AU636458B2 (en) Alginate hair setting compositions
AU8534198A (en) Derivatives of 2,5- and 3,5-disubstituted anilines, their preparation and use
AU6961896A (en) Herbicidal 3-(substituted benzoxazol-7-yl) and 3-(substituted benzothiazol-7-yl)-1-substituted-6-trifluoromethyl-2,4-(1h,3 h)pyrimidinediones
AU2942797A (en) Use of hydrophilic dispersion polymers for coated broke treatment
FI960507A0 (en) Redispersible, powdered core shell polymers, their preparation and use
MX9802962A (en) Keratin fibre treatment composition including at least one setting polymer and at least one ceramide-type compound, and methods
AU5626296A (en) Block copolymers, their preparation and their use as lubricants
EP0919576A4 (en) Novel copolymer, process for the preparation of the same, and use thereof
AU4493496A (en) Substituted 1,4-piperazine-heteroaryl derivatives as 5-ht1d receptor agonists
AU5168496A (en) Butyryl-tyrosinyl spermine, analogs thereof and methods of preparing and using same
AU6736596A (en) Prodrugs of 4-{3-(trans-3-dimethylaminocyclobutyl)-1h-indol-5-yl-methyl} -4(s)oxazolidin-2-one, their preparation and their use as 5ht1-like receptor agonists
AU5763396A (en) Benzothiazoles and benzoxazoles, as well as drugs containing them, their use and methods of preparing them
AU5331796A (en) Vectors for the transfection of eucaryotic cells, their use and target cells transfected thereby
AU9512298A (en) Beta3-adrenoreceptor agonists, agonist compositions and methods of using
HK1014938A1 (en) Oxazolidinone derivatives, their preparation and therapeutical use
AU4178497A (en) HTm4, methods of treatment and assays, agonists and antagonists
AU4994996A (en) Composition for the treatment of diarrhea, its use and its preparation
AU7135996A (en) Oxazolidin-2-one derivatives, preparation method therefor and therapeutical use thereof