AU2927492A - Phenol derivatives as agonists of a cyclic amp dependent protein kinase - Google Patents

Phenol derivatives as agonists of a cyclic amp dependent protein kinase

Info

Publication number
AU2927492A
AU2927492A AU29274/92A AU2927492A AU2927492A AU 2927492 A AU2927492 A AU 2927492A AU 29274/92 A AU29274/92 A AU 29274/92A AU 2927492 A AU2927492 A AU 2927492A AU 2927492 A AU2927492 A AU 2927492A
Authority
AU
Australia
Prior art keywords
compound
formula
group
hereinbefore defined
reacting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU29274/92A
Other languages
English (en)
Inventor
Kenneth John Murray
Roderick Alan Porter
Hunter Douglas Prain
Brian Herbert Warrington
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of AU2927492A publication Critical patent/AU2927492A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4021—Esters of aromatic acids (P-C aromatic linkage)

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AU29274/92A 1991-11-20 1992-11-16 Phenol derivatives as agonists of a cyclic amp dependent protein kinase Abandoned AU2927492A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9124579 1991-11-20
GB919124579A GB9124579D0 (en) 1991-11-20 1991-11-20 Chemical compounds

Publications (1)

Publication Number Publication Date
AU2927492A true AU2927492A (en) 1993-06-15

Family

ID=10704882

Family Applications (1)

Application Number Title Priority Date Filing Date
AU29274/92A Abandoned AU2927492A (en) 1991-11-20 1992-11-16 Phenol derivatives as agonists of a cyclic amp dependent protein kinase

Country Status (11)

Country Link
EP (1) EP0620815A1 (enrdf_load_stackoverflow)
JP (1) JPH07503235A (enrdf_load_stackoverflow)
AU (1) AU2927492A (enrdf_load_stackoverflow)
CA (1) CA2124003A1 (enrdf_load_stackoverflow)
GB (1) GB9124579D0 (enrdf_load_stackoverflow)
MX (1) MX9206709A (enrdf_load_stackoverflow)
NZ (1) NZ245168A (enrdf_load_stackoverflow)
PT (1) PT101073A (enrdf_load_stackoverflow)
TW (1) TW221812B (enrdf_load_stackoverflow)
WO (1) WO1993010107A1 (enrdf_load_stackoverflow)
ZA (1) ZA928894B (enrdf_load_stackoverflow)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3590082A (en) * 1967-10-06 1971-06-29 Merck & Co Inc 4-(p-fluorophenyl)salicylamide derivatives
EP0532531A1 (en) * 1990-05-21 1993-03-24 Smith Kline & French Laboratories Limited Phenol and pyridinol derivatives as pharmaceuticals

Also Published As

Publication number Publication date
GB9124579D0 (en) 1992-01-08
EP0620815A1 (en) 1994-10-26
PT101073A (pt) 1994-02-28
ZA928894B (en) 1994-05-18
JPH07503235A (ja) 1995-04-06
TW221812B (enrdf_load_stackoverflow) 1994-03-21
MX9206709A (es) 1993-05-01
WO1993010107A1 (en) 1993-05-27
NZ245168A (en) 1995-06-27
CA2124003A1 (en) 1993-05-27

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