AU2002251481A1 - Carboxylic acid derivative and salt thereof - Google Patents
Carboxylic acid derivative and salt thereofInfo
- Publication number
- AU2002251481A1 AU2002251481A1 AU2002251481A AU2002251481A AU2002251481A1 AU 2002251481 A1 AU2002251481 A1 AU 2002251481A1 AU 2002251481 A AU2002251481 A AU 2002251481A AU 2002251481 A AU2002251481 A AU 2002251481A AU 2002251481 A1 AU2002251481 A1 AU 2002251481A1
- Authority
- AU
- Australia
- Prior art keywords
- salt
- carboxylic acid
- acid derivative
- derivative
- carboxylic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001732 carboxylic acid derivatives Chemical class 0.000 title 1
- 150000001734 carboxylic acid salts Chemical class 0.000 title 1
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2001-123346 | 2001-04-20 | ||
JP2001123346 | 2001-04-20 | ||
JP2002-36274 | 2002-02-14 | ||
JP2002036274 | 2002-02-14 | ||
PCT/JP2002/003866 WO2002100812A1 (en) | 2001-04-20 | 2002-04-18 | Carboxylic acid derivative and salt thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002251481A1 true AU2002251481A1 (en) | 2003-05-15 |
AU2002251481B2 AU2002251481B2 (en) | 2007-08-09 |
Family
ID=26613950
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002251481A Ceased AU2002251481B2 (en) | 2001-04-20 | 2002-04-18 | Carboxylic acid derivative and salt thereof |
Country Status (19)
Country | Link |
---|---|
US (1) | US7544835B2 (en) |
EP (1) | EP1380562A4 (en) |
JP (1) | JP4131698B2 (en) |
KR (1) | KR100888001B1 (en) |
CN (1) | CN100522944C (en) |
AU (1) | AU2002251481B2 (en) |
BR (1) | BR0209027A (en) |
CA (1) | CA2442319C (en) |
CZ (1) | CZ20032727A3 (en) |
HU (1) | HUP0303810A3 (en) |
IL (1) | IL157731A0 (en) |
MX (1) | MXPA03009565A (en) |
NO (1) | NO329995B1 (en) |
NZ (2) | NZ528655A (en) |
PL (1) | PL206767B1 (en) |
RU (1) | RU2316537C2 (en) |
SG (1) | SG161743A1 (en) |
TW (1) | TWI311133B (en) |
WO (1) | WO2002100812A1 (en) |
Families Citing this family (54)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AUPO930697A0 (en) * | 1997-09-19 | 1997-10-09 | Walter And Eliza Hall Institute Of Medical Research, The | Catalytic antibodies and a method of producing same |
JP4256166B2 (en) * | 2001-03-28 | 2009-04-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | Carboxylic acid compound |
US7244861B2 (en) | 2001-03-30 | 2007-07-17 | Eisai Co., Ltd. | Benzene compound and salt thereof |
TWI311133B (en) | 2001-04-20 | 2009-06-21 | Eisai R&D Man Co Ltd | Carboxylic acid derivativeand the salt thereof |
EP1394147A4 (en) * | 2001-06-04 | 2007-10-24 | Eisai R&D Man Co Ltd | Carboxylic acid derivative and medicine comprising salt or ester of the same |
SK14912003A3 (en) * | 2001-06-07 | 2004-09-08 | Eli Lilly And Company | Receptor modulators activated by peroxizonal proliferators (PPAR) |
JPWO2003016265A1 (en) | 2001-08-17 | 2004-12-02 | エーザイ株式会社 | Cyclic compounds and PPAR agonists |
SE0104333D0 (en) | 2001-12-19 | 2001-12-19 | Astrazeneca Ab | Therapeutic agents |
US7816385B2 (en) * | 2002-12-20 | 2010-10-19 | High Point Pharmaceuticals, Llc | Dimeric dicarboxylic acid derivatives, their preparation and use |
JPWO2004082715A1 (en) * | 2003-03-20 | 2006-06-22 | エーザイ株式会社 | Concomitant medications as therapeutic agents for inflammatory bowel disease |
JP2007186515A (en) * | 2003-05-02 | 2007-07-26 | Takara Bio Inc | Curative agent |
MY150088A (en) * | 2003-05-19 | 2013-11-29 | Irm Llc | Immunosuppressant compounds and compositions |
GB0314131D0 (en) * | 2003-06-18 | 2003-07-23 | Astrazeneca Ab | Therapeutic agents |
JP4479656B2 (en) * | 2003-08-08 | 2010-06-09 | 宇部興産株式会社 | Alkynyl group-substituted fused heterocyclic compound, process for producing the same, and organic electroluminescence device using the same |
KR20060079798A (en) * | 2003-08-20 | 2006-07-06 | 액시스 파마슈티컬스 인코포레이티드 | Acetylene derivatives as inhibitors of histone deacetylase |
ES2433466T3 (en) | 2004-02-27 | 2013-12-11 | Amgen, Inc | Compounds, pharmaceutical compositions and methods for use in the treatment of metabolic disorders |
WO2005093423A2 (en) * | 2004-03-26 | 2005-10-06 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with peroxisome proliferative activated receptor alpha (ppara) |
JP4981662B2 (en) | 2004-05-05 | 2012-07-25 | ハイ・ポイント・ファーマスーティカルズ、エルエルシー | New compounds, their preparation and use |
JP2007536343A (en) | 2004-05-05 | 2007-12-13 | ノボ ノルディスク アクティーゼルスカブ | Phenoxyacetic acid derivatives as PPAR agonists |
FR2872159B1 (en) * | 2004-06-28 | 2007-10-05 | Merck Sante Soc Par Actions Si | NOVEL PHENYL CARBOXYLIC ACID DERIVATIVES AND THEIR USE IN THE TREATMENT OF DIABETES |
CA2571722C (en) * | 2004-07-01 | 2012-12-11 | F. Hoffmann-La Roche Ag | Phenyl derivatives comprising an acetylene group |
US7405236B2 (en) * | 2004-08-16 | 2008-07-29 | Hoffman-La Roche Inc. | Indole derivatives comprising an acetylene group |
ITMI20041825A1 (en) * | 2004-09-24 | 2004-12-24 | Medestea Res & Production Srl | RECEPTOR AGONISTS ACTIVATING THE PROLIFERATION OF PEROXYSOMES, USEFUL IN THE PREVENTION OR TREATMENT OF GASTRITIS |
US7816405B2 (en) * | 2005-04-19 | 2010-10-19 | Eisai R&D Management Co., Ltd. | Calcium bis [(2S)-3-[3-[(2S)-3-(4-chloro-2-cyanophenoxy)-2-fluoropropoxy]phenyl ]-2-isopropoxypropionate] and intermediate thereof |
KR20080007315A (en) * | 2005-04-19 | 2008-01-18 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | Calcium bis[(2s)-3-[3-[(2s)-3-(4-chloro-2-cyanophenoxy)-2-fluoropropoxy]phenyl]-2-isopropoxypropionate] and intermediate thereof |
US7465804B2 (en) | 2005-05-20 | 2008-12-16 | Amgen Inc. | Compounds, pharmaceutical compositions and methods for their use in treating metabolic disorders |
EP1893583B1 (en) | 2005-05-31 | 2012-04-04 | Pfizer Inc. | Substituted aryloxy-n-bicyclomethyl acetamide compounds as vr1 antagonists |
TW200718691A (en) * | 2005-06-10 | 2007-05-16 | Sigma Tau Ind Farmaceuti | Cinnamic and phenylpropiolic acid derivatives useful as anti-tumour agents |
BRPI0612730A2 (en) | 2005-06-30 | 2010-11-30 | Novo Nordisk As | compounds, their preparations and their use |
WO2007033002A1 (en) | 2005-09-14 | 2007-03-22 | Amgen Inc. | Conformationally constrained 3- (4-hydroxy-phenyl) - substituted-propanoic acids useful for treating metabolic disorders |
JP2007166908A (en) * | 2005-12-19 | 2007-07-05 | Sumitomo Chemical Co Ltd | Method for producing optically active 3-(3-hydroxyphenyl)-2-alkoxypropanoic acid or 3-(3-hydroxyphenyl)-2-alkoxypropanoic acid ester |
NZ568488A (en) | 2005-12-22 | 2011-07-29 | High Point Pharmaceuticals Llc | Phenoxy acetic acids as PPAR delta activators |
EP1999098A2 (en) | 2006-03-09 | 2008-12-10 | High Point Pharmaceuticals, LLC | Compounds that modulate ppar activity, their preparation and use |
SI2248812T1 (en) * | 2006-06-27 | 2014-04-30 | Takeda Pharmaceutical Company Limited | Fused cyclic compounds as gpr40 receptor modulators |
US7687526B2 (en) | 2006-09-07 | 2010-03-30 | Amgen Inc. | Benzo-fused compounds for use in treating metabolic disorders |
US7714008B2 (en) | 2006-09-07 | 2010-05-11 | Amgen Inc. | Heterocyclic GPR40 modulators |
BRPI0721424A2 (en) * | 2007-03-01 | 2014-03-25 | Bayer Schering Pharma Ag | RADIOFLUORATION METHODS |
EP2138484B1 (en) * | 2007-04-05 | 2015-08-26 | Daiichi Sankyo Company, Limited | Fused bicyclic heteroaryl derivatives |
ES2446419T3 (en) | 2007-04-16 | 2014-03-07 | Amgen, Inc | GPR40 modulators of substituted biphenylphenoxy, thiophenyl and aminophenylpropanoic acids |
NZ601866A (en) | 2007-06-29 | 2013-12-20 | Acucela Inc | Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders |
AU2008311355B2 (en) | 2007-10-10 | 2012-01-19 | Amgen Inc. | Substituted biphenyl GPR40 modulators |
JP2011515341A (en) | 2008-03-06 | 2011-05-19 | アムジエン・インコーポレーテツド | Conformationally restricted carboxylic acid derivatives useful for the treatment of metabolic disorders |
CA2739888C (en) | 2008-10-15 | 2013-11-19 | Amgen Inc. | Spirocyclic gpr40 modulators |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
EP2759533B1 (en) * | 2011-09-22 | 2017-08-02 | Takeda Pharmaceutical Company Limited | Condensed heterocyclic compound |
AU2013296187B2 (en) * | 2012-08-03 | 2016-09-29 | The Board Of Trustees Of The University Of Illinois | Enzyme-activating compounds and compositions |
CN109400502A (en) * | 2013-07-22 | 2019-03-01 | 新陈代谢解决方案开发公司 | The regulated compound of PPAR- for treating metabolic disease |
ES2784244T3 (en) * | 2013-12-18 | 2020-09-23 | Glaxosmithkline Ip Dev Ltd | Nrf2 regulators |
SI3240785T1 (en) | 2014-12-29 | 2021-11-30 | THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES, OFFICE OF TECHNOLOGY TRANSFER, NATIONAL INSTITUTES OF HEALTH | Small molecule inhibitors of lactate dehydrogenase and methods of use thereof |
CN108137557B (en) | 2015-06-15 | 2021-09-07 | 葛兰素史密斯克莱知识产权发展有限公司 | Nrf2 modulators |
LT3782996T (en) | 2015-06-15 | 2024-05-27 | Glaxosmithkline Intellectual Property Development Limited | Nrf2 regulators |
EP3359532A1 (en) | 2015-10-06 | 2018-08-15 | GlaxoSmithKline Intellectual Property Development Limited | Biaryl pyrazoles as nrf2 regulators |
Family Cites Families (41)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5649336A (en) | 1979-09-05 | 1981-05-02 | Glaxo Group Ltd | Phenol derivative* its manufacture and its use |
DE3026924A1 (en) * | 1980-07-16 | 1982-02-18 | Klinge Pharma GmbH & Co, 8000 München | 1,3-Di:phenoxy-propan-2-ol derivs. - used as hypolipaemics to reduce tri:glyceride and cholesterol levels in the blood |
JPS5764639A (en) * | 1980-10-04 | 1982-04-19 | Nippon Zoki Pharmaceut Co Ltd | Novel stilbene derivative, its preparation, and medical composition containing the same as active ingredent |
DE3682160D1 (en) | 1985-10-16 | 1991-11-28 | Merck Frosst Canada Inc | 2-SUBSTITUTED CHINOLINE. |
WO1989003819A1 (en) * | 1987-10-20 | 1989-05-05 | Otsuka Pharmaceutical Co., Ltd. | Phenylcarboxylic acid derivatives |
JPH02169584A (en) * | 1988-12-22 | 1990-06-29 | Mitsubishi Kasei Corp | Vinylthiazole derivative and drug containing same derivative as active ingredient |
NO179246C (en) * | 1991-11-20 | 1996-09-04 | Sankyo Co | Aromatic amino-alcohol derivatives and intermediates for their preparation |
NZ253742A (en) | 1992-07-03 | 1997-06-24 | Smithkline Beecham Plc | Heterocyclylaminoalkoxy substituted phenyl derivatives and pharmaceutical compositions |
GB9225386D0 (en) * | 1992-12-04 | 1993-01-27 | Smithkline Beecham Plc | Novel compounds |
GB9315148D0 (en) * | 1993-07-22 | 1993-09-08 | Smithkline Beecham Plc | Novel compounds |
JP3144624B2 (en) | 1995-06-02 | 2001-03-12 | 杏林製薬株式会社 | N-benzyldioxothiazolidylbenzamide derivative and method for producing the same |
EP1023907B1 (en) | 1997-07-24 | 2009-01-21 | Astellas Pharma Inc. | Medicinal compositions with cholesterol-lowering effect |
IL135177A0 (en) * | 1997-10-02 | 2001-05-20 | Sankyo Co | Amidocarboxylic acid derivatives and pharmaceutical compositions containing the same |
EA200000427A1 (en) | 1997-10-17 | 2001-02-26 | Авентис Фармасьютикалз Продактс Инк. | THERAPEUTIC APPLICATIONS OF QUINOLINE DERIVATIVES |
WO1999016758A1 (en) | 1997-10-27 | 1999-04-08 | Dr. Reddy's Research Foundation | Novel heterocyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them |
JPH11152269A (en) | 1997-11-20 | 1999-06-08 | Teijin Ltd | Biphenylamindine derivative |
MY153569A (en) | 1998-01-20 | 2015-02-27 | Mitsubishi Tanabe Pharma Corp | Inhibitors of ?4 mediated cell adhesion |
ATE274510T1 (en) | 1998-06-19 | 2004-09-15 | Chiron Corp | GLYCOGEN SYNTHASE KINASE 3 INHIBITORS |
FR2781222A1 (en) | 1998-07-17 | 2000-01-21 | Lipha | New cyclic peroxisome proliferator activated receptor activators, used to prevent or treat dyslipidemia, atherosclerosis and diabetes |
IL145922A0 (en) | 1999-04-28 | 2002-07-25 | Aventis Pharma Gmbh | Di-aryl acid derivatives as ppar receptor ligands |
PL351470A1 (en) * | 1999-04-28 | 2003-04-22 | Aventis Pharma Gmbh | Tri-aryl acid derivatives as ppar receptor ligands |
JP4618845B2 (en) | 1999-06-09 | 2011-01-26 | 杏林製薬株式会社 | Substituted phenylpropionic acid derivatives as human peroxisome proliferator-activated receptor (PPAR) alpha agonists |
CA2385083C (en) | 1999-09-17 | 2007-06-05 | Kyorin Pharmaceutical Co., Ltd. | O-anisamide derivatives |
TWI262185B (en) | 1999-10-01 | 2006-09-21 | Eisai Co Ltd | Carboxylic acid derivatives having anti-hyperglycemia and anti-hyperlipemia action, and pharmaceutical composition containing the derivatives |
DE19947457A1 (en) | 1999-10-02 | 2001-04-05 | Aventis Pharma Gmbh | New 2'-aminomethyl-biphenyl-2-carboxamide derivatives, are potassium channel blockers especially useful for treating re-entry or supraventricular arrhythmia or atrial fibrillation or flutter |
AR026414A1 (en) | 1999-11-10 | 2003-02-12 | Takeda Pharmaceutical | 5 MEMBER HETEROCICLICAL COMPUTERS CONTAINING NITROGEN |
JP2003520839A (en) * | 2000-01-28 | 2003-07-08 | ノボ ノルディスク アクティーゼルスカブ | New compounds, their production and use |
HUP0204574A3 (en) * | 2000-01-28 | 2003-08-28 | Novo Nordisk As | Propionic acid derivatives and their use in the treatment of diabetes and obesity, pharmaceutical compositions containing them and their preparation |
JP2001261612A (en) * | 2000-03-22 | 2001-09-26 | Mitsui Chemicals Inc | Catecholpropionic acid derivative and nuclear receptor agonist containing the same as active ingredient |
AU2001258838A1 (en) | 2000-05-29 | 2001-12-11 | Kyorin Pharmaceutical Co. Ltd. | Substituted phenylpropionic acid derivatives |
FR2812876B1 (en) | 2000-08-08 | 2002-09-27 | Galderma Res & Dev | NOVEL BIAROMATIC COMPOUNDS THAT ACTIVATE PPAR-GAMMA TYPE RECEPTORS AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS |
AU1339302A (en) | 2000-10-20 | 2002-05-06 | Biocryst Pharm Inc | Biaryl compounds as serine protease inhibitors |
EP1332131A2 (en) | 2000-11-07 | 2003-08-06 | Bristol-Myers Squibb Company | Acid derivatives useful as serine protease inhibitors |
JP4256166B2 (en) | 2001-03-28 | 2009-04-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | Carboxylic acid compound |
US7244861B2 (en) | 2001-03-30 | 2007-07-17 | Eisai Co., Ltd. | Benzene compound and salt thereof |
WO2002080899A1 (en) | 2001-03-30 | 2002-10-17 | Eisai Co., Ltd. | Remedial agent for digestive disease |
WO2002083616A1 (en) | 2001-04-10 | 2002-10-24 | Sankyo Company, Limited | α-SUBSTITUTED φ-ARYLFATTY ACID DERIVATIVE |
TWI311133B (en) | 2001-04-20 | 2009-06-21 | Eisai R&D Man Co Ltd | Carboxylic acid derivativeand the salt thereof |
EP1394147A4 (en) | 2001-06-04 | 2007-10-24 | Eisai R&D Man Co Ltd | Carboxylic acid derivative and medicine comprising salt or ester of the same |
JPWO2003016265A1 (en) | 2001-08-17 | 2004-12-02 | エーザイ株式会社 | Cyclic compounds and PPAR agonists |
FR2833949B1 (en) | 2001-12-21 | 2005-08-05 | Galderma Res & Dev | NOVEL PPARy RECEPTOR ACTIVATION LIGANDS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN HUMAN MEDICINE AND COSMETICS |
-
2002
- 2002-04-17 TW TW091107890A patent/TWI311133B/en not_active IP Right Cessation
- 2002-04-18 CZ CZ20032727A patent/CZ20032727A3/en unknown
- 2002-04-18 JP JP2003503583A patent/JP4131698B2/en not_active Expired - Fee Related
- 2002-04-18 MX MXPA03009565A patent/MXPA03009565A/en active IP Right Grant
- 2002-04-18 RU RU2003133744/04A patent/RU2316537C2/en not_active IP Right Cessation
- 2002-04-18 SG SG200608047-7A patent/SG161743A1/en unknown
- 2002-04-18 CN CNB028084985A patent/CN100522944C/en not_active Expired - Fee Related
- 2002-04-18 KR KR1020037013180A patent/KR100888001B1/en not_active IP Right Cessation
- 2002-04-18 BR BR0209027-9A patent/BR0209027A/en not_active Application Discontinuation
- 2002-04-18 EP EP02720489A patent/EP1380562A4/en not_active Withdrawn
- 2002-04-18 US US10/472,543 patent/US7544835B2/en not_active Expired - Fee Related
- 2002-04-18 PL PL367196A patent/PL206767B1/en not_active IP Right Cessation
- 2002-04-18 HU HU0303810A patent/HUP0303810A3/en unknown
- 2002-04-18 CA CA2442319A patent/CA2442319C/en not_active Expired - Fee Related
- 2002-04-18 NZ NZ528655A patent/NZ528655A/en unknown
- 2002-04-18 AU AU2002251481A patent/AU2002251481B2/en not_active Ceased
- 2002-04-18 NZ NZ539708A patent/NZ539708A/en unknown
- 2002-04-18 IL IL15773102A patent/IL157731A0/en unknown
- 2002-04-18 WO PCT/JP2002/003866 patent/WO2002100812A1/en active IP Right Grant
-
2003
- 2003-10-17 NO NO20034669A patent/NO329995B1/en not_active IP Right Cessation
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