AU2002248252B2 - Isoindole-imide compounds, compositions, and uses thereof - Google Patents

Isoindole-imide compounds, compositions, and uses thereof Download PDF

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Publication number
AU2002248252B2
AU2002248252B2 AU2002248252A AU2002248252A AU2002248252B2 AU 2002248252 B2 AU2002248252 B2 AU 2002248252B2 AU 2002248252 A AU2002248252 A AU 2002248252A AU 2002248252 A AU2002248252 A AU 2002248252A AU 2002248252 B2 AU2002248252 B2 AU 2002248252B2
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AU
Australia
Prior art keywords
alkyl
dioxo
piperidyl
methyl
aryl
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Ceased
Application number
AU2002248252A
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English (en)
Other versions
AU2002248252A1 (en
Inventor
Roger Shen-Chu Chen
Hon-Wah Man
George W. Muller
Michael J. Robarge
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Celgene Corp
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Celgene Corp
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Publication date
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of AU2002248252A1 publication Critical patent/AU2002248252A1/en
Priority to AU2006200717A priority Critical patent/AU2006200717B8/en
Application granted granted Critical
Publication of AU2002248252B2 publication Critical patent/AU2002248252B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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AU2002248252A 2000-12-27 2001-12-21 Isoindole-imide compounds, compositions, and uses thereof Ceased AU2002248252B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2006200717A AU2006200717B8 (en) 2000-12-27 2006-02-21 Isoindole-imide compounds, compositions, and uses thereof

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US25837200P 2000-12-27 2000-12-27
US60/258,372 2000-12-27
US09/972,487 2001-10-05
US09/972,487 US20030045552A1 (en) 2000-12-27 2001-10-05 Isoindole-imide compounds, compositions, and uses thereof
PCT/US2001/050401 WO2002059106A1 (en) 2000-12-27 2001-12-21 Isoindole-imide compounds, compositions, and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2006200717A Division AU2006200717B8 (en) 2000-12-27 2006-02-21 Isoindole-imide compounds, compositions, and uses thereof

Publications (2)

Publication Number Publication Date
AU2002248252A1 AU2002248252A1 (en) 2003-02-06
AU2002248252B2 true AU2002248252B2 (en) 2006-03-16

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Family Applications (3)

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AU2002248252A Ceased AU2002248252B2 (en) 2000-12-27 2001-12-21 Isoindole-imide compounds, compositions, and uses thereof
AU2006200717A Ceased AU2006200717B8 (en) 2000-12-27 2006-02-21 Isoindole-imide compounds, compositions, and uses thereof
AU2009202509A Ceased AU2009202509B2 (en) 2000-12-27 2009-06-23 Isoindole-imide compounds, compositions, and uses thereof

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AU2006200717A Ceased AU2006200717B8 (en) 2000-12-27 2006-02-21 Isoindole-imide compounds, compositions, and uses thereof
AU2009202509A Ceased AU2009202509B2 (en) 2000-12-27 2009-06-23 Isoindole-imide compounds, compositions, and uses thereof

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Country Link
US (1) US20030045552A1 (US20030045552A1-20030306-C00236.png)
EP (3) EP1363900B1 (US20030045552A1-20030306-C00236.png)
JP (3) JP4284071B2 (US20030045552A1-20030306-C00236.png)
KR (4) KR20070026879A (US20030045552A1-20030306-C00236.png)
AT (1) ATE352548T1 (US20030045552A1-20030306-C00236.png)
AU (3) AU2002248252B2 (US20030045552A1-20030306-C00236.png)
CA (1) CA2433021C (US20030045552A1-20030306-C00236.png)
CY (1) CY1106423T1 (US20030045552A1-20030306-C00236.png)
CZ (1) CZ20032041A3 (US20030045552A1-20030306-C00236.png)
DE (1) DE60126344T2 (US20030045552A1-20030306-C00236.png)
DK (1) DK1363900T3 (US20030045552A1-20030306-C00236.png)
ES (1) ES2275758T3 (US20030045552A1-20030306-C00236.png)
HK (1) HK1061396A1 (US20030045552A1-20030306-C00236.png)
HU (1) HU229003B1 (US20030045552A1-20030306-C00236.png)
IL (2) IL156646A0 (US20030045552A1-20030306-C00236.png)
MX (1) MXPA03005786A (US20030045552A1-20030306-C00236.png)
NZ (1) NZ526893A (US20030045552A1-20030306-C00236.png)
PT (1) PT1363900E (US20030045552A1-20030306-C00236.png)
WO (1) WO2002059106A1 (US20030045552A1-20030306-C00236.png)
ZA (1) ZA200305759B (US20030045552A1-20030306-C00236.png)

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US7629360B2 (en) * 1999-05-07 2009-12-08 Celgene Corporation Methods for the treatment of cachexia and graft v. host disease
US6458810B1 (en) 2000-11-14 2002-10-01 George Muller Pharmaceutically active isoindoline derivatives
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US11116782B2 (en) 2002-10-15 2021-09-14 Celgene Corporation Methods of treating myelodysplastic syndromes with a combination therapy using lenalidomide and azacitidine
US8404717B2 (en) * 2002-10-15 2013-03-26 Celgene Corporation Methods of treating myelodysplastic syndromes using lenalidomide
CN1326522C (zh) * 2002-10-24 2007-07-18 细胞基因公司 用于治疗、改变和控制疼痛的包含免疫调节化合物的组合物
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