ATE231510T1 - Penamsulfone als beta-laktamase inhibitoren - Google Patents

Penamsulfone als beta-laktamase inhibitoren

Info

Publication number
ATE231510T1
ATE231510T1 AT96924103T AT96924103T ATE231510T1 AT E231510 T1 ATE231510 T1 AT E231510T1 AT 96924103 T AT96924103 T AT 96924103T AT 96924103 T AT96924103 T AT 96924103T AT E231510 T1 ATE231510 T1 AT E231510T1
Authority
AT
Austria
Prior art keywords
beta
penamsulfones
lactamase inhibitors
antibiotics
lactamase
Prior art date
Application number
AT96924103T
Other languages
English (en)
Inventor
Samarendra Nath Maiti
Oludotun Adebayo Phillips
Andhe Venkat Narender Reddy
Eduardo Luis Setti
Ronald George Micetich
Chieko Kunugita
Fusahiro Higashitani
Akio Hyodo
Original Assignee
Naeja Pharmaceutical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Naeja Pharmaceutical Inc filed Critical Naeja Pharmaceutical Inc
Application granted granted Critical
Publication of ATE231510T1 publication Critical patent/ATE231510T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT96924103T 1995-08-04 1996-08-01 Penamsulfone als beta-laktamase inhibitoren ATE231510T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/511,227 US5686441A (en) 1995-08-04 1995-08-04 Penam sulfones as β-lactamase inhibitors
PCT/IB1996/000769 WO1997006172A1 (en) 1995-08-04 1996-08-01 Novel penam sulfones as beta-lactamase inhibitors

Publications (1)

Publication Number Publication Date
ATE231510T1 true ATE231510T1 (de) 2003-02-15

Family

ID=24033997

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96924103T ATE231510T1 (de) 1995-08-04 1996-08-01 Penamsulfone als beta-laktamase inhibitoren

Country Status (7)

Country Link
US (1) US5686441A (de)
EP (1) EP0842180B1 (de)
JP (1) JP2001509776A (de)
AT (1) ATE231510T1 (de)
CA (1) CA2228528A1 (de)
DE (1) DE69625910T2 (de)
WO (1) WO1997006172A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2812549B1 (fr) * 2000-08-03 2003-03-21 Aventis Pharma Sa Associations dalfopristine/quinupristine avec le cefpirome
CA2783572C (en) * 2005-12-07 2016-08-09 Basilea Pharmaceutica Ag Useful combinations of monobactam antibiotics with beta-lactamase inhibitors
AU2012233003B2 (en) * 2005-12-07 2014-12-18 Basilea Pharmaceutica Ag Useful combinations of monobactam antibiotics with beta-lactamase inhibitors
CN102161667B (zh) * 2011-05-05 2012-11-21 苏州二叶制药有限公司 磺苄西林钠及注射用磺苄西林钠
WO2013056163A1 (en) 2011-10-14 2013-04-18 The Regents Of The University Of California Beta-lactamase inhibitors
SI25892A (sl) * 2019-09-05 2021-03-31 Gorenje Gospodinjski Aparati, D.O.O. Pralni stroj, ki se polni s sprednje strani, z električnim svetlobnim telesom
EP4028404A4 (de) * 2019-09-11 2023-07-26 Tennor Therapeutics (Suzhou) Limited Penam-derivate zur behandlung bakterieller infektionen

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4562073A (en) * 1982-12-24 1985-12-31 Taiho Pharmaceutical Company Limited Penicillin derivatives
JPS6366187A (ja) * 1986-09-08 1988-03-24 Taiho Yakuhin Kogyo Kk 2α−置換ペニシリン誘導体
TW213460B (de) * 1991-02-15 1993-09-21 Hokuriku Pharmaceutical
EP0503597B1 (de) * 1991-03-13 1998-06-10 Otsuka Kagaku Kabushiki Kaisha Penamderivate und Verfahren zu deren Herstellung
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors

Also Published As

Publication number Publication date
US5686441A (en) 1997-11-11
CA2228528A1 (en) 1997-02-20
EP0842180A1 (de) 1998-05-20
WO1997006172A1 (en) 1997-02-20
JP2001509776A (ja) 2001-07-24
DE69625910T2 (de) 2003-11-06
EP0842180B1 (de) 2003-01-22
DE69625910D1 (de) 2003-02-27

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Legal Events

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