AT503764T - Inhibitors of the Hepatitis C virus - Google Patents

Inhibitors of the Hepatitis C virus

Info

Publication number
AT503764T
AT503764T AT03799806T AT03799806T AT503764T AT 503764 T AT503764 T AT 503764T AT 03799806 T AT03799806 T AT 03799806T AT 03799806 T AT03799806 T AT 03799806T AT 503764 T AT503764 T AT 503764T
Authority
AT
Austria
Prior art keywords
hepatitis
virus
inhibitors
Prior art date
Application number
AT03799806T
Other languages
German (de)
Inventor
Amy Ripka
Jeffrey Campbell
Andrew Good
Paul Scola
Ny Sin
Brian Venables
Original Assignee
Squibb Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US38215602P priority Critical
Application filed by Squibb Bristol Myers Co filed Critical Squibb Bristol Myers Co
Priority to PCT/US2003/015856 priority patent/WO2004032827A2/en
Publication of AT503764T publication Critical patent/AT503764T/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • C07K5/06165Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0821Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0823Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
AT03799806T 2002-05-20 2003-05-20 Inhibitors of the Hepatitis C virus AT503764T (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
US38215602P true 2002-05-20 2002-05-20
PCT/US2003/015856 WO2004032827A2 (en) 2002-05-20 2003-05-20 Hepatitis c virus inhibitors

Publications (1)

Publication Number Publication Date
AT503764T true AT503764T (en) 2011-04-15

Family

ID=32093711

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03799806T AT503764T (en) 2002-05-20 2003-05-20 Inhibitors of the Hepatitis C virus

Country Status (11)

Country Link
US (1) US7041698B2 (en)
EP (1) EP1506172B1 (en)
JP (1) JP4312718B2 (en)
AT (1) AT503764T (en)
AU (1) AU2003299519A1 (en)
DE (1) DE60336550D1 (en)
ES (1) ES2361011T3 (en)
IS (1) IS7533A (en)
NO (1) NO20044897L (en)
PL (1) PL215228B1 (en)
WO (1) WO2004032827A2 (en)

Families Citing this family (149)

* Cited by examiner, † Cited by third party
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JP4312718B2 (en) 2009-08-12
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EP1506172A4 (en) 2006-03-22
EP1506172B1 (en) 2011-03-30
ES2361011T3 (en) 2011-06-13
WO2004032827A3 (en) 2004-10-14
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WO2004032827A2 (en) 2004-04-22
AU2003299519A8 (en) 2004-05-04

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