AT467616T - Compounds with activity at the 11beta- hydroxasteroiddehydrogenase - Google Patents

Compounds with activity at the 11beta- hydroxasteroiddehydrogenase

Info

Publication number
AT467616T
AT467616T AT07102177T AT07102177T AT467616T AT 467616 T AT467616 T AT 467616T AT 07102177 T AT07102177 T AT 07102177T AT 07102177 T AT07102177 T AT 07102177T AT 467616 T AT467616 T AT 467616T
Authority
AT
Austria
Prior art keywords
hydroxasteroiddehydrogenase
11beta
activity
compounds
Prior art date
Application number
AT07102177T
Other languages
German (de)
Inventor
Anette Gundertofte
Anker Steen Jorgensen
Gita Camilla Tejlgaard Kampen
Henrik Sune Andersen
Inge Thoger Christensen
John Paul Kilburn
Original Assignee
High Point Pharmaceuticals Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to DKPA200300565 priority Critical
Priority to DKPA200300972 priority
Priority to DKPA200300990 priority
Priority to DKPA200300989 priority
Priority to DKPA200300988 priority
Priority to DKPA200300998 priority
Priority to DKPA200301910 priority
Priority to DKPA200400009 priority
Application filed by High Point Pharmaceuticals Llc filed Critical High Point Pharmaceuticals Llc
Publication of AT467616T publication Critical patent/AT467616T/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
AT07102177T 2003-04-11 2004-04-06 Compounds with activity at the 11beta- hydroxasteroiddehydrogenase AT467616T (en)

Priority Applications (8)

Application Number Priority Date Filing Date Title
DKPA200300565 2003-04-11
DKPA200300972 2003-06-27
DKPA200300990 2003-06-30
DKPA200300989 2003-06-30
DKPA200300988 2003-06-30
DKPA200300998 2003-07-02
DKPA200301910 2003-12-22
DKPA200400009 2004-01-06

Publications (1)

Publication Number Publication Date
AT467616T true AT467616T (en) 2010-05-15

Family

ID=36293394

Family Applications (2)

Application Number Title Priority Date Filing Date
AT04725891T AT482747T (en) 2003-04-11 2004-04-06 New amide derivatives and pharmaceutical uses
AT07102177T AT467616T (en) 2003-04-11 2004-04-06 Compounds with activity at the 11beta- hydroxasteroiddehydrogenase

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT04725891T AT482747T (en) 2003-04-11 2004-04-06 New amide derivatives and pharmaceutical uses

Country Status (6)

Country Link
US (1) US20090264414A1 (en)
EP (4) EP1618090A1 (en)
JP (2) JP4629657B2 (en)
AT (2) AT482747T (en)
DE (1) DE602004027171D1 (en)
WO (2) WO2004089896A1 (en)

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