AT426597T - Benzamid derivatives and their use as gluccoinase-activating agents - Google Patents

Benzamid derivatives and their use as gluccoinase-activating agents

Info

Publication number
AT426597T
AT426597T AT05708360T AT05708360T AT426597T AT 426597 T AT426597 T AT 426597T AT 05708360 T AT05708360 T AT 05708360T AT 05708360 T AT05708360 T AT 05708360T AT 426597 T AT426597 T AT 426597T
Authority
AT
Austria
Prior art keywords
gluccoinase
benzamid
derivatives
use
activating agents
Prior art date
Application number
AT05708360T
Other languages
German (de)
Inventor
Craig Johnstone
Darren Mckerrecher
Kurt Pike
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
Priority to GB0403593A priority Critical patent/GB0403593D0/en
Priority to GB0413386A priority patent/GB0413386D0/en
Priority to GB0423039A priority patent/GB0423039D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34890799&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AT426597(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of AT426597T publication Critical patent/AT426597T/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • C07D231/40Acylated on said nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/44Acylated amino or imino radicals
    • C07D277/46Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
AT05708360T 2004-02-18 2005-02-15 Benzamid derivatives and their use as gluccoinase-activating agents AT426597T (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
GB0403593A GB0403593D0 (en) 2004-02-18 2004-02-18 Compounds
GB0413386A GB0413386D0 (en) 2004-06-16 2004-06-16 Compounds
GB0423039A GB0423039D0 (en) 2004-10-16 2004-10-16 Compounds

Publications (1)

Publication Number Publication Date
AT426597T true AT426597T (en) 2009-04-15

Family

ID=34890799

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05708360T AT426597T (en) 2004-02-18 2005-02-15 Benzamid derivatives and their use as gluccoinase-activating agents

Country Status (18)

Country Link
US (2) US20080280872A1 (en)
EP (2) EP1718624B1 (en)
JP (1) JP2007523142A (en)
KR (1) KR20070007103A (en)
AR (1) AR047678A1 (en)
AT (1) AT426597T (en)
AU (1) AU2005214132B9 (en)
BR (1) BRPI0507746A (en)
CA (1) CA2554310A1 (en)
DE (1) DE602005013491D1 (en)
ES (1) ES2322709T3 (en)
HK (1) HK1096092A1 (en)
IL (1) IL177216D0 (en)
NO (1) NO20063452L (en)
RU (1) RU2392275C2 (en)
TW (1) TW200602028A (en)
UY (1) UY28756A1 (en)
WO (1) WO2005080359A1 (en)

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BRPI0516595A (en) * 2004-10-16 2008-09-23 Astrazeneca Ab process for making a compound, and, compound
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TW200714597A (en) * 2005-05-27 2007-04-16 Astrazeneca Ab Chemical compounds
NZ575514A (en) * 2005-07-09 2009-11-27 Astrazeneca Ab Heteroaryl benzamide derivatives for use as GLK activators in the treatment of diabetes
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TW200738621A (en) * 2005-11-28 2007-10-16 Astrazeneca Ab Chemical process
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WO2008012227A2 (en) 2006-07-24 2008-01-31 F. Hoffmann-La Roche Ag Pyrazoles as glucokinase activators
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WO2010082601A1 (en) * 2009-01-16 2010-07-22 第一三共株式会社 Novel 2,5-disubstituted pyrrole derivative
GB0902434D0 (en) * 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
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AR076220A1 (en) 2009-04-09 2011-05-26 Astrazeneca Ab Pyrazole derivatives [4,5 - e] pyrimidine
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Also Published As

Publication number Publication date
AR047678A1 (en) 2006-02-01
CA2554310A1 (en) 2005-09-01
DE602005013491D1 (en) 2009-05-07
RU2392275C2 (en) 2010-06-20
EP1718624B1 (en) 2009-03-25
KR20070007103A (en) 2007-01-12
IL177216D0 (en) 2006-12-10
AU2005214132A1 (en) 2005-09-01
NO20063452L (en) 2006-10-31
UY28756A1 (en) 2005-09-30
WO2005080359A1 (en) 2005-09-01
AU2005214132B2 (en) 2009-05-07
ES2322709T3 (en) 2009-06-25
EP2048137A1 (en) 2009-04-15
US20110034432A1 (en) 2011-02-10
US20080280872A1 (en) 2008-11-13
TW200602028A (en) 2006-01-16
HK1096092A1 (en) 2009-09-11
RU2006130684A (en) 2008-03-27
BRPI0507746A (en) 2007-07-10
AU2005214132B9 (en) 2009-06-25
EP1718624A1 (en) 2006-11-08
JP2007523142A (en) 2007-08-16

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