AT414508T - Solid pharmaceutical pharmaceutical forms using a s1p receptor agonist and a sugar alcohol - Google Patents

Solid pharmaceutical pharmaceutical forms using a s1p receptor agonist and a sugar alcohol

Info

Publication number
AT414508T
AT414508T AT04725895T AT04725895T AT414508T AT 414508 T AT414508 T AT 414508T AT 04725895 T AT04725895 T AT 04725895T AT 04725895 T AT04725895 T AT 04725895T AT 414508 T AT414508 T AT 414508T
Authority
AT
Austria
Prior art keywords
pharmaceutical
receptor agonist
sugar alcohol
s1p receptor
solid pharmaceutical
Prior art date
Application number
AT04725895T
Other languages
German (de)
Inventor
Tomoyuki Oomura
Madhusudhan Pudipeddi
Alan Royce
Colleen Ruegger
Masaki Sasaki
Tokuhiro Tamura
Original Assignee
Novartis Pharma Gmbh
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
Priority to US46121503P priority Critical
Application filed by Novartis Pharma Gmbh, Mitsubishi Pharma Corp filed Critical Novartis Pharma Gmbh
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32326722&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AT414508(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of AT414508T publication Critical patent/AT414508T/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/145Amines having sulfur, e.g. thiurams (>N—C(S)—S—C(S)—N< and >N—C(S)—S—S—C(S)—N<), Sulfinylamines (—N=SO), Sulfonylamines (—N=SO2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
AT04725895T 2003-04-08 2004-04-06 Solid pharmaceutical pharmaceutical forms using a s1p receptor agonist and a sugar alcohol AT414508T (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
US46121503P true 2003-04-08 2003-04-08

Publications (1)

Publication Number Publication Date
AT414508T true AT414508T (en) 2008-12-15

Family

ID=32326722

Family Applications (3)

Application Number Title Priority Date Filing Date
AT04725895T AT414508T (en) 2003-04-08 2004-04-06 Solid pharmaceutical pharmaceutical forms using a s1p receptor agonist and a sugar alcohol
ATA606/2004A AT501681B1 (en) 2003-04-08 2004-04-06 Solid oral pharmaceutical composition containing 2-amino-1,3-propandiole
AT0074408A AT504853A2 (en) 2003-04-08 2008-05-08 Organic connections

Family Applications After (2)

Application Number Title Priority Date Filing Date
ATA606/2004A AT501681B1 (en) 2003-04-08 2004-04-06 Solid oral pharmaceutical composition containing 2-amino-1,3-propandiole
AT0074408A AT504853A2 (en) 2003-04-08 2008-05-08 Organic connections

Country Status (43)

Country Link
US (9) US20060275357A1 (en)
EP (5) EP2319502A1 (en)
JP (3) JP5495467B2 (en)
KR (3) KR101367574B1 (en)
CN (2) CN1767819B (en)
AR (3) AR043987A1 (en)
AT (3) AT414508T (en)
AU (1) AU2004228929B2 (en)
BE (1) BE1015972A5 (en)
BR (1) BRPI0409250A (en)
CA (2) CA2707750A1 (en)
CL (2) CL2004000745A1 (en)
CY (2) CY1110260T1 (en)
DE (4) DE122011100047I1 (en)
DK (2) DK1613288T3 (en)
EC (1) ECSP056090A (en)
ES (3) ES2556947T3 (en)
FR (1) FR2854073B1 (en)
GB (1) GB2400318B (en)
GR (1) GR1005052B (en)
HK (3) HK1071685A1 (en)
HR (3) HRP20050886B1 (en)
HU (2) HUE028247T2 (en)
IE (1) IE20040246A1 (en)
IL (3) IL170888A (en)
IS (2) IS2682B (en)
IT (1) ITMI20040682A1 (en)
LU (1) LU91867I9 (en)
MA (1) MA27729A1 (en)
MX (1) MXPA05010860A (en)
MY (1) MY141249A (en)
NO (4) NO329332B1 (en)
NZ (3) NZ592339A (en)
PE (5) PE20150676A1 (en)
PL (2) PL1613288T3 (en)
PT (1) PT1613288E (en)
RU (5) RU2358716C2 (en)
SG (1) SG175449A1 (en)
SI (2) SI1613288T1 (en)
TN (1) TNSN05256A1 (en)
TW (1) TWI332847B (en)
WO (1) WO2004089341A1 (en)
ZA (1) ZA200507394B (en)

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Also Published As

Publication number Publication date
CY1110260T1 (en) 2014-04-09
RU2010146697A (en) 2012-05-27
PT1613288E (en) 2009-02-25
NO20055231D0 (en) 2005-11-07
EP2008650A2 (en) 2008-12-31
GR20040100121A (en) 2004-12-17
GB2400318B (en) 2005-08-10
CA2521325A1 (en) 2004-10-21
HUS1100016I1 (en) 2016-08-29
ES2228282A1 (en) 2005-04-01
PL1613288T3 (en) 2009-07-31
CA2707750A1 (en) 2004-10-21
AT501681A1 (en) 2006-10-15
EP2316431A1 (en) 2011-05-04
IL242037D0 (en) 2015-11-30
AR078781A2 (en) 2011-11-30
NO20131287L (en) 2006-01-09
ECSP056090A (en) 2006-03-01
RU2475237C2 (en) 2013-02-20
JP5495467B2 (en) 2014-05-21
CN1767819A (en) 2006-05-03
GB0407819D0 (en) 2004-05-12
JP2013177404A (en) 2013-09-09
GB2400318A (en) 2004-10-13
TNSN05256A1 (en) 2007-07-10
ES2320767T3 (en) 2009-05-28
IL197578A (en) 2015-10-29
EP1613288A1 (en) 2006-01-11
AR078782A2 (en) 2011-11-30
NO335120B1 (en) 2014-09-22
SI2316431T1 (en) 2016-04-29
EP1613288B1 (en) 2008-11-19
US20060275357A1 (en) 2006-12-07
AR043987A1 (en) 2005-08-17
TWI332847B (en) 2010-11-11
US20130108675A1 (en) 2013-05-02
US20140011885A1 (en) 2014-01-09
NO2011016I1 (en) 2011-09-19
ITMI20040682A1 (en) 2004-07-06
HK1091114A1 (en) 2009-06-26
NZ586280A (en) 2011-12-22
SG175449A1 (en) 2011-11-28
PE20050396A1 (en) 2005-07-05
LU91867I2 (en) 2011-11-08
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