AR192370A1 - Procedimiento para la obtencion de derivados de piridazina - Google Patents
Procedimiento para la obtencion de derivados de piridazinaInfo
- Publication number
- AR192370A1 AR192370A1 AR242634A AR24263472A AR192370A1 AR 192370 A1 AR192370 A1 AR 192370A1 AR 242634 A AR242634 A AR 242634A AR 24263472 A AR24263472 A AR 24263472A AR 192370 A1 AR192370 A1 AR 192370A1
- Authority
- AR
- Argentina
- Prior art keywords
- procedure
- obtaining
- pyridazine derivatives
- pyridazine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/20—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB2873771 | 1971-06-18 | ||
FR7219096A FR2141697B1 (es) | 1971-06-18 | 1972-05-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR192370A1 true AR192370A1 (es) | 1973-02-14 |
Family
ID=26217112
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR242634A AR192370A1 (es) | 1971-06-18 | 1972-06-19 | Procedimiento para la obtencion de derivados de piridazina |
Country Status (13)
Country | Link |
---|---|
US (1) | US4169158A (es) |
JP (1) | JPS5550943B1 (es) |
AR (1) | AR192370A1 (es) |
AU (1) | AU472247B2 (es) |
BE (1) | BE784727A (es) |
CA (1) | CA1003833A (es) |
CH (1) | CH546769A (es) |
DE (1) | DE2229215C2 (es) |
ES (1) | ES403998A1 (es) |
FR (1) | FR2141697B1 (es) |
GB (1) | GB1345880A (es) |
NL (1) | NL177893C (es) |
SE (1) | SE392899B (es) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2510998B1 (fr) * | 1981-08-07 | 1986-01-10 | Sanofi Sa | Nouveaux derives amines de la pyridazine, leur procede de preparation et les medicaments, a action desinhibitrice, qui en comportent |
FR2510997A1 (fr) * | 1981-08-10 | 1983-02-11 | Sanofi Sa | Nouveaux derives de la methyl-4 phenyl-6 pyridazine, procede pour leur preparation et medicaments actifs sur le systeme nerveux central en contenant |
FR2511366A1 (fr) * | 1981-08-11 | 1983-02-18 | Sanofi Sa | Nouveaux derives de la pyridazine, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent |
FR2539741A1 (fr) * | 1983-01-21 | 1984-07-27 | Sanofi Sa | Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent |
FR2539739B1 (fr) * | 1983-01-24 | 1985-11-22 | Sanofi Sa | Nouveaux derives de la naphtyl pyridazine actifs sur le systeme nerveux central, procede de preparation de ces derives et medicaments en contenant |
FR2539742B1 (fr) * | 1983-01-24 | 1986-09-05 | Sanofi Sa | Derives amines de la pyridazine substitues en position 6 par un heterocycle ou un alicycle, lesdits derives etant actifs sur le systeme nerveux central |
CA1218655A (en) * | 1983-01-28 | 1987-03-03 | Kathleen Biziere | Process for the preparation of pyridazine derivatives having a psychotropic action |
FR2555178B1 (fr) * | 1983-11-18 | 1986-04-18 | Sanofi Sa | Derives cyanes de la pyridazine ayant une action psychotrope, leur mode de preparation et les medicaments en contenant |
FR2540115B1 (fr) * | 1983-01-28 | 1985-06-07 | Sanofi Sa | Derive de la pyridazine ayant une action psychotrope, son mode de preparation et les medicaments en contenant |
FR2625201B1 (fr) * | 1987-12-24 | 1990-06-15 | Sanofi Sa | Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant |
US5461053A (en) * | 1989-02-07 | 1995-10-24 | Sanofi | Pyridazine derivatives |
PT93060B (pt) | 1989-02-07 | 1995-12-29 | Sanofi Sa | Processo para a obtencao de derivados de piridazina e de composicoes farmaceuticas que os contem |
FR2642757B1 (fr) * | 1989-02-07 | 1991-05-24 | Sanofi Sa | Nouveaux derives de la pyridazine, procede de preparation et compositions pharmaceutiques en contenant |
FR2642648B1 (fr) * | 1989-02-07 | 1991-06-21 | Sanofi Sa | Utilisation de derives d'alkyl-5 pyridazine comme medicaments actifs sur le systeme cholinergique |
FR2642754B1 (fr) * | 1989-02-07 | 1991-05-24 | Sanofi Sa | Nouveaux derives de la pyridazine, procede de preparation et compositions pharmaceutiques en contenant |
US20100210590A1 (en) * | 1995-09-27 | 2010-08-19 | Northwestern University | Compositions and treatments for seizure-related disorders |
WO2003018563A1 (en) * | 2001-08-31 | 2003-03-06 | Northwestern University | Anti-inflammatory and protein kinase inhibitor composition and method of use |
WO2006050389A2 (en) | 2004-11-02 | 2006-05-11 | Northwestern University | Pyridazine compounds, compositions and methods |
CA2589102C (en) | 2004-11-02 | 2013-08-13 | Northwestern University | Pyridazine compounds and methods for using the compounds to treat inflammatory diseases |
BRPI0613564A2 (pt) | 2005-07-04 | 2011-01-18 | Novo Nordisk As | compostos, seus usos na preparação de composições farmacêuticas e composições farmacêuticas compreendendo os mesmos |
RU2442775C2 (ru) * | 2005-07-04 | 2012-02-20 | Хай Пойнт Фармасьютикалс, ЛЛС | Антагонисты гистаминовых н3-рецепторов |
WO2007127474A2 (en) | 2006-04-28 | 2007-11-08 | Northwestern University | Compositions and treatments using pyridazine compounds and cholinesterase inhibitors |
WO2007127448A2 (en) * | 2006-04-28 | 2007-11-08 | Northwestern University | Salts of pyridazine compounds |
BRPI0710938A2 (pt) | 2006-04-28 | 2012-06-26 | Univ Northwestern | formulações contendo compostos de piridazina para o tratamento de doenças neuroinflamatórias |
CA2653062A1 (en) | 2006-05-23 | 2007-11-29 | Transtech Pharma, Inc. | 6- (4-cyclopropylpiperazin-1-yl) -2 ' -methyl- [3, 4 ' ] -bipyridine and its use as a medicament |
AU2007267197B2 (en) | 2006-05-29 | 2011-12-01 | High Point Pharmaceuticals, Llc | 3- (1, 3-Benzodioxol-5-yl) -6- (4-cyclopropylpiperazin-1-yl) -pyridazine, its salts and solvates and its use as histamine H3 receptor antagonist |
EP2014656A3 (en) | 2007-06-11 | 2011-08-24 | High Point Pharmaceuticals, LLC | New heteocyclic h3 antagonists |
EP2291181B9 (en) | 2008-04-18 | 2013-09-11 | University College Dublin National University Of Ireland, Dublin | Captodiamine for the treatment of depression symptoms |
AR081331A1 (es) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos |
AR081626A1 (es) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos |
US9133123B2 (en) | 2010-04-23 | 2015-09-15 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
CN112041679A (zh) | 2018-01-23 | 2020-12-04 | 古斯塔夫·鲁西研究所 | 米那普利用于降低肿瘤生长的用途 |
-
1971
- 1971-06-18 GB GB2873771A patent/GB1345880A/en not_active Expired
-
1972
- 1972-05-29 FR FR7219096A patent/FR2141697B1/fr not_active Expired
- 1972-06-12 BE BE784727A patent/BE784727A/xx not_active IP Right Cessation
- 1972-06-12 CA CA144,468A patent/CA1003833A/en not_active Expired
- 1972-06-15 DE DE2229215A patent/DE2229215C2/de not_active Expired
- 1972-06-16 SE SE7207999A patent/SE392899B/xx unknown
- 1972-06-16 AU AU43500/72A patent/AU472247B2/en not_active Expired
- 1972-06-16 CH CH903672A patent/CH546769A/fr not_active IP Right Cessation
- 1972-06-17 ES ES403998A patent/ES403998A1/es not_active Expired
- 1972-06-19 AR AR242634A patent/AR192370A1/es active
- 1972-06-19 NL NLAANVRAGE7208355,A patent/NL177893C/xx not_active IP Right Cessation
- 1972-06-19 JP JP6054172A patent/JPS5550943B1/ja active Pending
-
1977
- 1977-07-29 US US05/820,489 patent/US4169158A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
US4169158A (en) | 1979-09-25 |
AU4350072A (en) | 1973-12-20 |
GB1345880A (en) | 1974-02-06 |
JPS5550943B1 (es) | 1980-12-20 |
AU472247B2 (en) | 1973-12-20 |
CH546769A (fr) | 1974-03-15 |
FR2141697B1 (es) | 1976-09-17 |
NL7208355A (es) | 1972-12-20 |
NL177893C (nl) | 1985-12-16 |
FR2141697A1 (es) | 1973-01-26 |
DE2229215C2 (de) | 1984-09-06 |
ES403998A1 (es) | 1975-06-01 |
BE784727A (fr) | 1972-10-02 |
CA1003833A (en) | 1977-01-18 |
DE2229215A1 (de) | 1973-01-25 |
SE392899B (sv) | 1977-04-25 |
NL177893B (nl) | 1985-07-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR192370A1 (es) | Procedimiento para la obtencion de derivados de piridazina | |
AR193462A1 (es) | Procedimiento para la preparacion de derivados de cetona | |
AR199879A1 (es) | Procedimiento para la elaboracion de 4-aza-benzimidazoles | |
AR200387A1 (es) | Procedimiento para preparar derivados de trifluorometilfenilpiperazina | |
AR203002A1 (es) | Procedimiento para la preparacion de derivados de tetrahidrodibenzo-imidazo-azepinas | |
AR192765A1 (es) | Procedimiento para la preparacion de derivados de la fenil-3-tiourea | |
AR199084A1 (es) | Procedimiento para la obtencion de derivados 2-nitroimidazol | |
AR192914A1 (es) | Procedimiento para la obtencion de compuesto yodoetinilicos | |
AR209571A1 (es) | Procedimiento para preparar compuestos derivados de fluorenona | |
AR195785A1 (es) | Procedimiento para la preparacion de derivados de benzocicloheptaisoquinolina | |
AR204899A1 (es) | Procedimiento para la preparacion de 3-carbamoiloximetilcefalosporinas | |
AR192732A1 (es) | Procedimiento para la preparacion de derivados de guanidinofenilurea | |
AR196408A1 (es) | Procedimiento para la preparacion de derivados de tienodiazepina | |
AR203017A1 (es) | Procedimiento para la preparacion de fenilimidazolidinonas | |
AR199605A1 (es) | Procedimiento para preparar dihidro-2aminoisoquinolinas | |
AR205784A1 (es) | Procedimiento para la elaboracion de penicilamina | |
AR209254A1 (es) | Procedimiento para la preparacion de derivados de fenil-bencilcetona | |
AR200859A1 (es) | Procedimiento para la obtencion de nuevos derivados de diazepina | |
AR193576A1 (es) | Procedimiento para la preparacion de pirimidotriacinas | |
AR209577A1 (es) | Procedimiento para la obtencion de 1-fenoxi-3-amino-propan-2-ol-n-sustituido | |
AR197007A1 (es) | Procedimiento para la preparacion de sulfonilaminopirimidinas | |
AR198166A1 (es) | Procedimiento para la obtencion de derivados de piridina | |
AR203728A1 (es) | Procedimiento para la preparacion de derivados de nitropirazol | |
AR208273A1 (es) | Procedimiento para la preparacion de derivados de nitroquinazolinona | |
AR203192A1 (es) | Procedimiento para la obtencion de nuevos derivados de diazepina |