AR061620A1 - Suspensiones acuosas de tmc278 - Google Patents

Suspensiones acuosas de tmc278

Info

Publication number
AR061620A1
AR061620A1 ARP070102777A ARP070102777A AR061620A1 AR 061620 A1 AR061620 A1 AR 061620A1 AR P070102777 A ARP070102777 A AR P070102777A AR P070102777 A ARP070102777 A AR P070102777A AR 061620 A1 AR061620 A1 AR 061620A1
Authority
AR
Argentina
Prior art keywords
tmc278
pharmaceutical compositions
suspensions
waterproof
waterproof suspensions
Prior art date
Application number
ARP070102777A
Other languages
English (en)
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38833797&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR061620(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of AR061620A1 publication Critical patent/AR061620A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Composiciones farmacéuticas para la administracion por inyeccion intramuscular o subcutánea, que comprende micro- o nanopartículas del compuesto NNRTI TMC278, suspendido en un portador acuoso farmacéuticamente aceptable, el uso de dichas composiciones farmacéuticas en el tratamiento y la prevencion de infeccion por VIH y proceso para preparar dicha composicion.
ARP070102777A 2006-06-23 2007-06-22 Suspensiones acuosas de tmc278 AR061620A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06115938 2006-06-23

Publications (1)

Publication Number Publication Date
AR061620A1 true AR061620A1 (es) 2008-09-10

Family

ID=38833797

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070102777A AR061620A1 (es) 2006-06-23 2007-06-22 Suspensiones acuosas de tmc278

Country Status (32)

Country Link
US (4) US20090176813A1 (es)
EP (2) EP2040671B1 (es)
JP (1) JP5292288B2 (es)
KR (1) KR101406879B1 (es)
CN (1) CN101478950B (es)
AP (1) AP2618A (es)
AR (1) AR061620A1 (es)
AU (1) AU2007262941B2 (es)
BR (2) BR122020011487B1 (es)
CA (1) CA2654115C (es)
CL (1) CL2007001847A1 (es)
CY (1) CY1120564T1 (es)
DK (1) DK2040671T3 (es)
EA (1) EA021700B1 (es)
ES (1) ES2662068T3 (es)
HR (1) HRP20180629T1 (es)
HU (1) HUE038797T2 (es)
IL (1) IL195491A (es)
JO (1) JOP20200160A1 (es)
LT (1) LT2040671T (es)
MX (1) MX2009000158A (es)
NZ (1) NZ573291A (es)
PE (1) PE20080210A1 (es)
PL (1) PL2040671T3 (es)
PT (1) PT2040671T (es)
RS (1) RS57111B1 (es)
SG (1) SG173315A1 (es)
SI (1) SI2040671T1 (es)
TW (1) TWI413521B (es)
UA (1) UA97641C2 (es)
UY (1) UY30431A1 (es)
WO (1) WO2007147882A2 (es)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
TWI457136B (zh) * 2005-04-04 2014-10-21 Tibotec Pharm Ltd Hiv-感染之預防
AR065720A1 (es) 2007-03-14 2009-06-24 Tibotec Pharm Ltd Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso.
EP2306980A2 (en) * 2008-06-30 2011-04-13 Tibotec Pharmaceuticals Powders for reconstitution
SG172398A1 (en) * 2008-12-24 2011-07-28 Tibotec Pharm Ltd Implantable devices for treating hiv
DK2696848T3 (da) 2011-04-15 2020-10-12 Janssen Pharmaceutica Nv Frysetørrede nanosuspensioner af lægemiddel
JO3387B1 (ar) 2011-12-16 2019-03-13 Glaxosmithkline Llc مشتقات بيتولين
WO2014093941A1 (en) 2012-12-14 2014-06-19 Glaxosmithkline Llc Pharmaceutical compositions
JP2017528497A (ja) * 2014-09-26 2017-09-28 グラクソスミスクライン、インテレクチュアル、プロパティー、(ナンバー2)、リミテッドGlaxosmithkline Intellectual Property (No.2) Limited 長時間作用型医薬組成物
WO2017209732A1 (en) * 2016-05-31 2017-12-07 Taimed Biologics, Inc. A long acting pharmaceutical composition of protease inhibitor
TWI678203B (zh) * 2016-05-31 2019-12-01 中裕新藥股份有限公司 蛋白酶抑制劑之長效醫藥組合物
US10369129B2 (en) * 2016-05-31 2019-08-06 Taimed Biologics, Inc. Long acting pharmaceutical composition of protease inhibitor
HRP20240118T1 (hr) 2016-10-24 2024-04-12 Janssen Sciences Ireland Unlimited Company Disperzivni pripravci
PE20200336A1 (es) 2017-07-14 2020-02-14 Janssen Pharmaceutica Nv Formulaciones a largo plazo
CN113440529B (zh) * 2020-03-25 2023-11-14 江苏恒瑞医药股份有限公司 一种可注射的药物组合物及其制备方法
WO2022008644A1 (en) 2020-07-09 2022-01-13 Janssen Pharmaceutica Nv Long-acting formulations
CA3182854A1 (en) 2020-07-09 2022-01-13 Rene Holm Long-acting formulations
CN115867259A (zh) 2020-07-09 2023-03-28 詹森药业有限公司 长效配制品
WO2022109555A1 (en) 2020-11-17 2022-05-27 Janssen Sciences Ireland Unlimited Company Treatment or prevention of hiv infection
MX2023005760A (es) * 2020-11-17 2023-07-31 Janssen Sciences Ireland Unlimited Co Tratamiento o prevención de una enfermedad o trastorno.
WO2023088964A1 (en) 2021-11-17 2023-05-25 Janssen Sciences Ireland Unlimited Company Dissolution test
TW202408516A (zh) 2022-04-22 2024-03-01 愛爾蘭商健生科學愛爾蘭無限公司 液體組成物
TW202406551A (zh) 2022-04-22 2024-02-16 愛爾蘭商健生科學愛爾蘭無限公司 冷凍乾燥組成物(一)
WO2023222754A1 (en) 2022-05-17 2023-11-23 Janssen Sciences Ireland Unlimited Company Rilpivirine for use in the treatment or prevention of hiv infection
TW202408527A (zh) 2022-05-17 2024-03-01 愛爾蘭商健生科學愛爾蘭無限公司 治療或預防hiv感染(二)
WO2024068699A1 (en) 2022-09-28 2024-04-04 Janssen Pharmaceutica Nv Long-acting formulations
WO2024068693A1 (en) 2022-09-28 2024-04-04 Janssen Pharmaceutica Nv Long-acting formulations

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US4102124A (en) * 1976-07-12 1978-07-25 Swager William E Locking clevis or the like
US5145684A (en) 1991-01-25 1992-09-08 Sterling Drug Inc. Surface modified drug nanoparticles
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JP5324098B2 (ja) * 2004-11-16 2013-10-23 アルケルメス ファーマ アイルランド リミテッド 注射可能なナノ粒子のオランザピン製剤
TWI457136B (zh) * 2005-04-04 2014-10-21 Tibotec Pharm Ltd Hiv-感染之預防
EA014914B1 (ru) * 2006-01-20 2011-02-28 Тиботек Фармасьютикалз Лтд. Долговременное лечение вич-инфекции

Also Published As

Publication number Publication date
CL2007001847A1 (es) 2008-02-08
EA200970047A1 (ru) 2009-04-28
CN101478950B (zh) 2013-02-06
MX2009000158A (es) 2009-01-23
US20220273653A1 (en) 2022-09-01
JP2009541271A (ja) 2009-11-26
JOP20200160A1 (ar) 2022-10-30
EP2040671B1 (en) 2018-01-24
UA97641C2 (en) 2012-03-12
SG173315A1 (en) 2011-08-29
AU2007262941B2 (en) 2013-11-21
EA021700B1 (ru) 2015-08-31
PE20080210A1 (es) 2008-04-11
AU2007262941A1 (en) 2007-12-27
SI2040671T1 (en) 2018-05-31
BRPI0713334B1 (pt) 2024-02-20
EP3366278B1 (en) 2024-08-07
NZ573291A (en) 2011-11-25
IL195491A (en) 2014-11-30
RS57111B1 (sr) 2018-06-29
US20150010637A1 (en) 2015-01-08
EP3366278A1 (en) 2018-08-29
IL195491A0 (en) 2009-09-01
UY30431A1 (es) 2008-01-31
HUE038797T2 (hu) 2018-11-28
PL2040671T3 (pl) 2018-08-31
BRPI0713334A8 (pt) 2018-01-02
BRPI0713334A2 (pt) 2012-03-06
CA2654115C (en) 2015-12-22
US11389447B2 (en) 2022-07-19
EP2040671A2 (en) 2009-04-01
US20090176813A1 (en) 2009-07-09
BR122020011487B1 (pt) 2024-02-20
US20160089369A1 (en) 2016-03-31
CA2654115A1 (en) 2007-12-27
TW200817008A (en) 2008-04-16
TWI413521B (zh) 2013-11-01
JP5292288B2 (ja) 2013-09-18
AP2008004682A0 (en) 2008-12-31
CY1120564T1 (el) 2019-07-10
HRP20180629T1 (hr) 2018-06-01
PT2040671T (pt) 2018-03-14
WO2007147882A3 (en) 2008-06-19
WO2007147882A2 (en) 2007-12-27
LT2040671T (lt) 2018-05-10
AP2618A (en) 2013-03-18
ES2662068T3 (es) 2018-04-05
KR20090023703A (ko) 2009-03-05
DK2040671T3 (en) 2018-05-07
CN101478950A (zh) 2009-07-08
KR101406879B1 (ko) 2014-06-13

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