AR054782A2 - Composiciones farmaceuticas y tabletas que contienen irbesartan en combinacion con un diuretico - Google Patents

Composiciones farmaceuticas y tabletas que contienen irbesartan en combinacion con un diuretico

Info

Publication number
AR054782A2
AR054782A2 ARP060102579A ARP060102579A AR054782A2 AR 054782 A2 AR054782 A2 AR 054782A2 AR P060102579 A ARP060102579 A AR P060102579A AR P060102579 A ARP060102579 A AR P060102579A AR 054782 A2 AR054782 A2 AR 054782A2
Authority
AR
Argentina
Prior art keywords
diuretic
irbesartan
combination
pharmaceutical compositions
tablets containing
Prior art date
Application number
ARP060102579A
Other languages
English (en)
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23876256&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR054782(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of AR054782A2 publication Critical patent/AR054782A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Abstract

Composiciones farmacéuticas que contienen irbesartan en combinacion con un diurético, y que proveen tabletas que contienen una elevada cantidad de agente activo y que gozan de excelentes propiedades de humectacion y desintegracion. Reivindicacion 1: Una composicion farmacéutica, caracterizada porque comprende basado en peso: (a) 20 a 70 %, de irbesartan o una de sus sales farmacéuticamente aceptables; (b) 2 a 33 %, de diurético, siendo la carga combinada de (a) y (b), no superior al 85%; (c), 1 a 70 %, de diluyente; (d) 2 a 20 %, de ligante; (e) 1 a 10 %, de desintegrante, (f) 0,1 a 5 % de antiadherente; y (g) 0,2 a 5 % de lubricante, uno o mas excipientes farmacéuticamente aceptables, en donde una tableta formada a partir de dicha composicion tiene una velocidad de disolucion tal que aproximadamente de 80 % o más, del irbesartan o de sus sales del mismo, contenido en dicha tableta, se disuelve en el lapso de 30 minutos.
ARP060102579A 1995-06-07 2006-06-16 Composiciones farmaceuticas y tabletas que contienen irbesartan en combinacion con un diuretico AR054782A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US47261895A 1995-06-07 1995-06-07

Publications (1)

Publication Number Publication Date
AR054782A2 true AR054782A2 (es) 2007-07-18

Family

ID=23876256

Family Applications (2)

Application Number Title Priority Date Filing Date
AR10297996A AR002350A1 (es) 1995-06-07 1996-06-06 Composiciones farmacéuticas que contienen irbesartan
ARP060102579A AR054782A2 (es) 1995-06-07 2006-06-16 Composiciones farmaceuticas y tabletas que contienen irbesartan en combinacion con un diuretico

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR10297996A AR002350A1 (es) 1995-06-07 1996-06-06 Composiciones farmacéuticas que contienen irbesartan

Country Status (23)

Country Link
EP (2) EP0747050B2 (es)
JP (1) JP3162626B2 (es)
KR (1) KR100442719B1 (es)
CN (1) CN1149083C (es)
AR (2) AR002350A1 (es)
AT (2) ATE503478T1 (es)
AU (1) AU702651B2 (es)
CA (1) CA2177772C (es)
CZ (1) CZ291532B6 (es)
DE (2) DE69638348D1 (es)
DK (2) DK0747050T4 (es)
ES (2) ES2205000T5 (es)
HK (1) HK1002384A1 (es)
HU (1) HU229369B1 (es)
IL (1) IL118309A (es)
NO (2) NO310495B1 (es)
NZ (2) NZ329547A (es)
PL (1) PL184893B1 (es)
PT (2) PT747050E (es)
RU (2) RU2181590C2 (es)
SG (1) SG49956A1 (es)
TW (1) TW442301B (es)
ZA (1) ZA964337B (es)

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JP2018009032A (ja) * 2017-10-19 2018-01-18 大原薬品工業株式会社 化学的な安定性が向上したイルベサルタン含有錠剤
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Also Published As

Publication number Publication date
EP1275391A1 (en) 2003-01-15
ATE248594T1 (de) 2003-09-15
DE69629755D1 (de) 2003-10-09
NO310495B1 (no) 2001-07-16
SG49956A1 (en) 1998-06-15
HU229369B1 (en) 2013-11-28
IL118309A0 (en) 1996-09-12
AU702651B2 (en) 1999-02-25
AU5476396A (en) 1996-12-19
HUP9601564A2 (hu) 1998-09-28
PT747050E (pt) 2003-12-31
RU2001130903A (ru) 2004-02-27
RU2210368C1 (ru) 2003-08-20
HK1002384A1 (en) 1998-08-21
NO20004743L (no) 1996-12-09
NZ286612A (en) 1998-03-25
CA2177772A1 (en) 1996-12-08
ES2205000T5 (es) 2013-05-30
AR002350A1 (es) 1998-03-11
PL314670A1 (en) 1996-12-09
NO962387L (no) 1996-12-09
JPH08333253A (ja) 1996-12-17
ES2205000T3 (es) 2004-05-01
NO20004743D0 (no) 2000-09-22
NO310393B1 (no) 2001-07-02
EP0747050A1 (en) 1996-12-11
NZ329547A (en) 1998-06-26
HU9601564D0 (en) 1996-08-28
EP0747050B2 (en) 2013-02-13
CA2177772C (en) 2007-04-10
CZ163496A3 (en) 1996-12-11
NO962387D0 (no) 1996-06-06
DE69629755T3 (de) 2013-08-08
KR970000232A (ko) 1997-01-21
CN1144656A (zh) 1997-03-12
IL118309A (en) 2003-06-24
DK0747050T4 (da) 2013-05-21
DK1275391T3 (da) 2011-07-11
ZA964337B (en) 1997-11-28
ATE503478T1 (de) 2011-04-15
DK0747050T3 (da) 2003-12-15
KR100442719B1 (ko) 2004-10-08
EP1275391B1 (en) 2011-03-30
HUP9601564A3 (en) 2000-12-28
TW442301B (en) 2001-06-23
PL184893B1 (pl) 2003-01-31
PT1275391E (pt) 2011-06-30
MX9602103A (es) 1997-09-30
ES2363127T3 (es) 2011-07-21
JP3162626B2 (ja) 2001-05-08
DE69629755T2 (de) 2004-07-01
CZ291532B6 (cs) 2003-03-12
EP0747050B1 (en) 2003-09-03
RU2181590C2 (ru) 2002-04-27
CN1149083C (zh) 2004-05-12
DE69638348D1 (de) 2011-05-12

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