AR045997A1 - Composiciones farmaceuticas estables que contienen derivados de azetidina - Google Patents

Composiciones farmaceuticas estables que contienen derivados de azetidina

Info

Publication number
AR045997A1
AR045997A1 ARP040102495A ARP040102495A AR045997A1 AR 045997 A1 AR045997 A1 AR 045997A1 AR P040102495 A ARP040102495 A AR P040102495A AR P040102495 A ARP040102495 A AR P040102495A AR 045997 A1 AR045997 A1 AR 045997A1
Authority
AR
Argentina
Prior art keywords
azetidine
solid
composition
semi
composition according
Prior art date
Application number
ARP040102495A
Other languages
English (en)
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of AR045997A1 publication Critical patent/AR045997A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Inorganic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Sistemas semi-sólidos que contienen derivados de azetidina. Formulaciones de derivados de azetidina para administración oral. Reivindicación 1: Una composición faramcéutica estable que comprende al menos un derivado de azetidina de fórmula general 1a o 2b, en un sistema que comprende un material semisólido polimérico qu es vitamina E TPGS(R). Reivindicación 6: Un proceso para preparar una composición de acuerdo con una de las reivindicaciones 1 a 5, en el que, cuando es apropiado, se prepara la mexcla de los excipientes principales, después de claentar, si feura necesario, en el caso de excipientes sólidos o semisólidos y después, si fuera necesario, la mezcla con los aditivos adicionales, y después se anade el derivado de azetidina como se ha definido en la reivindicación 1 y cuando sea apropiado, el ingrediente activo que puede potenciar los efectos del derivado de azetidina de fórmula general (1a) o (1b), definido en la reivindicación 1, y se mantiene la agitación para obtener una mezcla homogénea. Reivindicación7: Un kit de presentación que contiene una composición de acuerdo con la reivindicación 1 o 2 y una composición que comprende un ingrediente activo que puede potenciar los efectos del derivad de azetidina definido en la reivindicación 1. Reivindicación 9: Un kit de presentanción que contiene una composición de acuerdo con la reivindicación 1 o 2 y una composición que comprende un agente que activa la neurotransmisión dopaminérgica en el cerebro.
ARP040102495A 2003-07-18 2004-07-15 Composiciones farmaceuticas estables que contienen derivados de azetidina AR045997A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03291796A EP1498122A1 (en) 2003-07-18 2003-07-18 Semi-solid systems containing azetidine derivatives

Publications (1)

Publication Number Publication Date
AR045997A1 true AR045997A1 (es) 2005-11-23

Family

ID=33462259

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP040102495A AR045997A1 (es) 2003-07-18 2004-07-15 Composiciones farmaceuticas estables que contienen derivados de azetidina

Country Status (30)

Country Link
US (2) US20050026898A1 (es)
EP (2) EP1498122A1 (es)
JP (1) JP2009513560A (es)
KR (1) KR20060040691A (es)
CN (1) CN1822831A (es)
AR (1) AR045997A1 (es)
AU (1) AU2004262498B2 (es)
BR (1) BRPI0412737A (es)
CA (1) CA2532669A1 (es)
CR (1) CR8179A (es)
EC (1) ECSP066292A (es)
GT (1) GT200400135A (es)
HR (1) HRP20060022A2 (es)
IL (1) IL173111A0 (es)
MA (1) MA27922A1 (es)
MX (1) MXPA06000483A (es)
MY (1) MY142077A (es)
NO (1) NO20060509L (es)
OA (1) OA13191A (es)
PA (1) PA8606701A1 (es)
PE (1) PE20050287A1 (es)
RS (1) RS20060016A (es)
RU (1) RU2343915C2 (es)
SG (1) SG144141A1 (es)
TN (1) TNSN06013A1 (es)
TW (1) TW200522945A (es)
UA (1) UA80633C2 (es)
UY (1) UY28421A1 (es)
WO (1) WO2005013973A1 (es)
ZA (1) ZA200600490B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2007123366A (ru) * 2004-11-24 2008-12-27 Мерк Энд Ко. Жидкие и полутвердые фармацевтические препаративные формы для перорального введения замещенного амида
FR2923719B1 (fr) * 2007-11-15 2009-11-20 Sanofi Aventis Compositions pharmaceutiques a base de derives d'azetidine
CN101926757B (zh) * 2010-09-01 2013-01-02 北京大学 一种难溶性药物的液体组合物及其制备方法
JP5868414B2 (ja) * 2010-11-08 2016-02-24 カディラ ファーマシューティカルズ リミテッド タキソイドの医薬組成物
CN105848643A (zh) * 2013-12-23 2016-08-10 强生消费者公司 消旋卡多曲组合物

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996036316A1 (en) * 1995-05-19 1996-11-21 Abbott Laboratories Self-emulsifying formulations of lipophilic drugs
EP1015046A2 (en) * 1998-07-14 2000-07-05 Em Industries, Inc. Microdisperse drug delivery systems
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
US6355631B1 (en) * 2000-03-03 2002-03-12 Aventis Pharma S.A. Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and their preparation
FR2814678B1 (fr) * 2000-10-04 2002-12-20 Aventis Pharma Sa Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite
FR2829027A1 (fr) * 2001-08-29 2003-03-07 Aventis Pharma Sa Association avec un antagoniste du recepteur cb1, les compositions pharmaceutiques les contenant et leur utilisation pour le traitement de la maladie de parkinson
FR2833842B1 (fr) * 2001-12-21 2004-02-13 Aventis Pharma Sa Compositions pharmaceutiques a base de derives d'azetidine
EP1498123A1 (en) * 2003-07-18 2005-01-19 Aventis Pharma S.A. Emulsifying systems containing azetidine derivatives

Also Published As

Publication number Publication date
AU2004262498A2 (en) 2005-02-17
CR8179A (es) 2006-09-22
AU2004262498A1 (en) 2005-02-17
RU2343915C2 (ru) 2009-01-20
US20080293686A1 (en) 2008-11-27
BRPI0412737A (pt) 2006-09-26
TW200522945A (en) 2005-07-16
AU2004262498B2 (en) 2009-01-22
NO20060509L (no) 2006-01-31
RS20060016A (en) 2008-06-05
MXPA06000483A (es) 2006-04-05
OA13191A (en) 2006-12-13
TNSN06013A1 (en) 2007-10-03
EP1498122A1 (en) 2005-01-19
PE20050287A1 (es) 2005-06-13
GT200400135A (es) 2005-08-25
ECSP066292A (es) 2006-10-25
PA8606701A1 (es) 2005-02-04
IL173111A0 (en) 2006-06-11
MY142077A (en) 2010-08-30
SG144141A1 (en) 2008-07-29
UY28421A1 (es) 2005-02-28
RU2006105011A (ru) 2006-06-10
KR20060040691A (ko) 2006-05-10
US20050026898A1 (en) 2005-02-03
WO2005013973A1 (en) 2005-02-17
UA80633C2 (en) 2007-10-10
HRP20060022A2 (en) 2006-02-28
CN1822831A (zh) 2006-08-23
ZA200600490B (en) 2007-05-30
EP1648442A1 (en) 2006-04-26
MA27922A1 (fr) 2006-06-01
CA2532669A1 (en) 2005-02-17
JP2009513560A (ja) 2009-04-02

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal