AP201609180A0 - 4-{4-[(1 e)-4-(2,9-diazaspiro[5.5]undec-2-yl)but-1 -en-1 -yl]-2-methylbenzyl}-5-(propan-2-yl)-1 h-pyrazol-3-yl beta-d- glucopyranoside acetate - Google Patents

4-{4-[(1 e)-4-(2,9-diazaspiro[5.5]undec-2-yl)but-1 -en-1 -yl]-2-methylbenzyl}-5-(propan-2-yl)-1 h-pyrazol-3-yl beta-d- glucopyranoside acetate

Info

Publication number
AP201609180A0
AP201609180A0 AP201609180A AP201609180A AP201609180A0 AP 201609180 A0 AP201609180 A0 AP 201609180A0 AP 201609180 A AP201609180 A AP 201609180A AP 201609180 A AP201609180 A AP 201609180A AP 201609180 A0 AP201609180 A0 AP 201609180A0
Authority
AP
ARIPO
Prior art keywords
yl
diazaspiro
undec
methylbenzyl
pyrazol
Prior art date
Application number
AP201609180A
Inventor
Reutzel-Edens Susan Marie
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US201361901488P priority Critical
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Priority to PCT/US2014/063161 priority patent/WO2015069541A1/en
Publication of AP201609180A0 publication Critical patent/AP201609180A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
AP201609180A 2013-11-08 2014-10-30 4-{4-[(1 e)-4-(2,9-diazaspiro[5.5]undec-2-yl)but-1 -en-1 -yl]-2-methylbenzyl}-5-(propan-2-yl)-1 h-pyrazol-3-yl beta-d- glucopyranoside acetate AP201609180A0 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
US201361901488P true 2013-11-08 2013-11-08
PCT/US2014/063161 WO2015069541A1 (en) 2013-11-08 2014-10-30 4-{4-[(1 e)-4-(2,9-diazaspiro[5.5]undec-2-yl)but-1 -en-1 -yl]-2-methylbenzyl}-5-(propan-2-yl)-1 h-pyrazol-3-yl beta-d- glucopyranoside acetate

Publications (1)

Publication Number Publication Date
AP201609180A0 true AP201609180A0 (en) 2016-04-30

Family

ID=51982747

Family Applications (1)

Application Number Title Priority Date Filing Date
AP201609180A AP201609180A0 (en) 2013-11-08 2014-10-30 4-{4-[(1 e)-4-(2,9-diazaspiro[5.5]undec-2-yl)but-1 -en-1 -yl]-2-methylbenzyl}-5-(propan-2-yl)-1 h-pyrazol-3-yl beta-d- glucopyranoside acetate

Country Status (31)

Country Link
US (1) US9573970B2 (en)
EP (1) EP3066108B1 (en)
JP (1) JP6197113B2 (en)
KR (1) KR101858881B1 (en)
CN (1) CN105705509B (en)
AP (1) AP201609180A0 (en)
AR (1) AR098670A1 (en)
AU (1) AU2014347065B2 (en)
CA (1) CA2925128C (en)
CL (1) CL2016000791A1 (en)
CR (1) CR20160165A (en)
DK (1) DK3066108T3 (en)
DO (1) DOP2016000067A (en)
EA (1) EA028801B1 (en)
ES (1) ES2703944T3 (en)
HR (1) HRP20182061T1 (en)
IL (1) IL244899D0 (en)
LT (1) LT3066108T (en)
MA (1) MA39019A1 (en)
MX (1) MX2016005999A (en)
NZ (1) NZ718118A (en)
PE (1) PE08842016A1 (en)
PH (1) PH12016500851A1 (en)
PL (1) PL3066108T3 (en)
RS (1) RS58050B1 (en)
SI (1) SI3066108T1 (en)
SV (1) SV2016005190A (en)
TN (1) TN2016000112A1 (en)
TW (1) TWI655198B (en)
UA (1) UA118767C2 (en)
WO (1) WO2015069541A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018231691A1 (en) * 2017-06-12 2018-12-20 Lignamed, Llc Process for the preparation of (s,s)-secoisolariciresinol diglucoside and (r,r)-secoisolariciresinol diglucoside

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1213296E (en) 1999-08-31 2004-08-31 Kissei Pharmaceutical Derivatives of glucopiranosiloxipirazole medical compositions that contain them and intermediaries in their production
DE60230591D1 (en) 2001-02-26 2009-02-12 Kissei Pharmaceutical Glykopyranosyloxypyrazolderivate and their medical use
CA2448741C (en) 2001-05-30 2010-06-22 Kissei Pharmaceutical Co., Ltd. Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
ZA200501094B (en) * 2002-08-08 2006-10-25 Kissei Pharmaceutical Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof
CA2494179C (en) * 2002-08-08 2012-04-24 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof
JP2004137245A (en) 2002-08-23 2004-05-13 Kissei Pharmaceut Co Ltd Pyrazole derivative, pharmaceutical composition containing the same, its pharmaceutical use and production intermediate
DE102004028241B4 (en) 2004-06-11 2007-09-13 Sanofi-Aventis Deutschland Gmbh New fluoroglycoside pyrazoles, pharmaceutical compositions containing these compounds and manufacture of these drugs
BRPI0711949A2 (en) * 2006-05-19 2012-01-17 Taisho Pharma Co Ltd phenyl-compound and glycitol
ES2548578T3 (en) 2007-12-27 2015-10-19 Kissei Pharmaceutical Co., Ltd. Monosebacato of a pyrazole derivative
US8466113B2 (en) 2009-02-23 2013-06-18 Taisho Pharmaceutical Co., Ltd. 4-isopropylphenyl glucitol compounds as SGLT1 inhibitors
WO2011039338A2 (en) 2009-10-02 2011-04-07 Sanofi-Aventis Use of compounds with sglt-1/sglt-2 inhibitor activity for producing medicaments for treatment of bone diseases
US8163704B2 (en) 2009-10-20 2012-04-24 Novartis Ag Glycoside derivatives and uses thereof
JO3136B1 (en) * 2012-05-10 2017-09-20 Lilly Co Eli Pyrazole compounds as sglt1 inhibitors

Also Published As

Publication number Publication date
CN105705509B (en) 2018-12-04
LT3066108T (en) 2019-01-25
PE08842016A1 (en) 2016-09-10
EP3066108A1 (en) 2016-09-14
JP6197113B2 (en) 2017-09-13
AU2014347065A1 (en) 2016-04-07
PL3066108T3 (en) 2019-03-29
EA028801B1 (en) 2017-12-29
SI3066108T1 (en) 2018-12-31
WO2015069541A1 (en) 2015-05-14
CA2925128C (en) 2017-10-17
HRP20182061T1 (en) 2019-02-08
EA201690749A1 (en) 2016-08-31
CN105705509A (en) 2016-06-22
TN2016000112A1 (en) 2017-07-05
IL244899D0 (en) 2016-05-31
CL2016000791A1 (en) 2016-11-11
NZ718118A (en) 2017-11-24
RS58050B1 (en) 2019-02-28
TWI655198B (en) 2019-04-01
DOP2016000067A (en) 2016-04-15
AU2014347065B2 (en) 2016-09-29
MA39019A1 (en) 2017-04-28
AR098670A1 (en) 2016-06-08
JP2016539099A (en) 2016-12-15
CA2925128A1 (en) 2015-05-14
PH12016500851A1 (en) 2016-06-20
SV2016005190A (en) 2018-11-01
KR101858881B1 (en) 2018-05-16
MX2016005999A (en) 2016-07-22
CR20160165A (en) 2016-06-08
ES2703944T3 (en) 2019-03-13
KR20160067157A (en) 2016-06-13
DK3066108T3 (en) 2019-01-02
US20160215011A1 (en) 2016-07-28
EP3066108B1 (en) 2018-10-24
UA118767C2 (en) 2019-03-11
TW201609783A (en) 2016-03-16
US9573970B2 (en) 2017-02-21

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