AP201407762A0 - New forms and salts of a dihydropyrrolo[1,2C]imidazolyl aldosterone synthase or aromatase inhibitor - Google Patents

New forms and salts of a dihydropyrrolo[1,2C]imidazolyl aldosterone synthase or aromatase inhibitor

Info

Publication number
AP201407762A0
AP201407762A0 AP201407762A AP201407762A AP201407762A0 AP 201407762 A0 AP201407762 A0 AP 201407762A0 AP 201407762 A AP201407762 A AP 201407762A AP 201407762 A AP201407762 A AP 201407762A AP 201407762 A0 AP201407762 A0 AP 201407762A0
Authority
AP
ARIPO
Prior art keywords
dihydropyrrolo
imidazolyl
2c
salts
aromatase inhibitor
Prior art date
Application number
AP201407762A
Inventor
Paul Sutton
Eric Loeser
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US201261587280P priority Critical
Application filed by Novartis Ag filed Critical Novartis Ag
Priority to PCT/US2013/021521 priority patent/WO2013109514A1/en
Publication of AP201407762A0 publication Critical patent/AP201407762A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
AP201407762A 2012-01-17 2013-01-15 New forms and salts of a dihydropyrrolo[1,2C]imidazolyl aldosterone synthase or aromatase inhibitor AP201407762A0 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
US201261587280P true 2012-01-17 2012-01-17
PCT/US2013/021521 WO2013109514A1 (en) 2012-01-17 2013-01-15 New forms and salts of a dihydropyrrolo[1,2-c]imidazolyl aldosterone synthase or aromatase inhibitor

Publications (1)

Publication Number Publication Date
AP201407762A0 true AP201407762A0 (en) 2014-07-31

Family

ID=47604250

Family Applications (1)

Application Number Title Priority Date Filing Date
AP201407762A AP201407762A0 (en) 2012-01-17 2013-01-15 New forms and salts of a dihydropyrrolo[1,2C]imidazolyl aldosterone synthase or aromatase inhibitor

Country Status (39)

Country Link
US (2) US9334276B2 (en)
EP (1) EP2804863B1 (en)
JP (1) JP5749410B2 (en)
KR (2) KR20140141687A (en)
CN (1) CN104039793B (en)
AP (1) AP201407762A0 (en)
AR (1) AR089728A1 (en)
AU (1) AU2013209952B2 (en)
BR (1) BR112014017260A8 (en)
CA (1) CA2863339A1 (en)
CL (1) CL2014001863A1 (en)
CO (1) CO7000775A2 (en)
CR (1) CR20140345A (en)
CU (1) CU20140086A7 (en)
CY (1) CY1117914T1 (en)
DK (1) DK2804863T3 (en)
EA (1) EA026232B1 (en)
ES (1) ES2564143T3 (en)
GT (1) GT201400155A (en)
HK (1) HK1198536A1 (en)
HR (1) HRP20160178T1 (en)
HU (1) HUE026984T2 (en)
IL (1) IL233541A (en)
IN (1) IN2014DN06781A (en)
JO (1) JO3137B1 (en)
MA (1) MA35858B1 (en)
MX (1) MX2014008686A (en)
NZ (1) NZ626277A (en)
PE (1) PE23582014A1 (en)
PH (1) PH12014501638A1 (en)
RS (1) RS54589B1 (en)
SG (1) SG11201404061YA (en)
SM (1) SMT201600083B (en)
TN (1) TN2014000256A1 (en)
TW (1) TWI609869B (en)
UA (1) UA114803C2 (en)
UY (1) UY34576A (en)
WO (1) WO2013109514A1 (en)
ZA (1) ZA201404314B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ601077A (en) * 2010-01-14 2014-07-25 Novartis Ag Use of an adrenal hormone-modifying agent
EP2815749A1 (en) 2013-06-20 2014-12-24 IP Gesellschaft für Management mbH Solid form of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione having specified X-ray diffraction pattern
PL3166596T3 (en) * 2014-07-07 2018-11-30 Novartis Ag Pharmaceutical dosage forms
CA2973539A1 (en) 2015-01-29 2016-08-04 Novartis Ag Process for the production of condensed imidazolo derivatives
WO2016164476A2 (en) * 2015-04-06 2016-10-13 Millendo Therapeutics, Inc. Combination therapy for treating disorders associated with excess cortisol production
WO2018078049A1 (en) * 2016-10-27 2018-05-03 Damian Pharma Ag Aldosterone synthase inhibitor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4617307A (en) * 1984-06-20 1986-10-14 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridine derivatives as aromatase inhibitors
US5066656A (en) 1989-11-01 1991-11-19 Janssen Pharmaceutica N.V. Pharmacologically active (6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-5-yl)- and (5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-5-yl) substituted 1H-benzotriazole derivatives
MTP1076B (en) * 1990-01-12 1991-09-30 Ciba Geigy Ag Hemihydrate
AU668708B2 (en) 1992-01-27 1996-05-16 Janssen Pharmaceutica N.V. Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
PT1565463E (en) * 2002-11-18 2008-09-10 Novartis Ag Imidazo[1,5a] pyridine derivatives and methods for treating aldosterone mediated diseases
GT200600381A (en) 2005-08-25 2007-03-28 organic compounds
MX2009006481A (en) 2006-12-18 2009-06-26 Novartis Ag Organic compounds.
US8575160B2 (en) 2009-11-30 2013-11-05 Novartis Ag Imidazole derivatives as aldosterone synthase inhibitors
NZ601077A (en) 2010-01-14 2014-07-25 Novartis Ag Use of an adrenal hormone-modifying agent

Also Published As

Publication number Publication date
KR20140141687A (en) 2014-12-10
MX2014008686A (en) 2014-08-27
EP2804863B1 (en) 2015-12-02
KR20140093726A (en) 2014-07-28
CO7000775A2 (en) 2014-07-21
SMT201600083B (en) 2016-04-29
BR112014017260A2 (en) 2017-06-13
CN104039793B (en) 2017-05-10
PH12014501638A1 (en) 2014-10-13
AU2013209952A1 (en) 2014-07-24
JP5749410B2 (en) 2015-07-15
TN2014000256A1 (en) 2015-09-30
CR20140345A (en) 2014-09-09
US20160176883A1 (en) 2016-06-23
BR112014017260A8 (en) 2017-07-04
EA201491374A1 (en) 2014-12-30
US20140364470A1 (en) 2014-12-11
HUE026984T2 (en) 2016-08-29
MA35858B1 (en) 2014-12-01
JO3137B1 (en) 2017-09-20
IL233541A (en) 2018-12-31
CU20140086A7 (en) 2014-12-26
ES2564143T3 (en) 2016-03-18
CN104039793A (en) 2014-09-10
IL233541D0 (en) 2014-08-31
DK2804863T3 (en) 2016-03-07
SI2804863T1 (en) 2016-05-31
CY1117914T1 (en) 2017-05-17
CL2014001863A1 (en) 2014-11-07
HRP20160178T1 (en) 2016-03-25
UY34576A (en) 2013-09-02
UA114803C2 (en) 2017-08-10
PH12014501638B1 (en) 2014-10-13
HK1198536A1 (en) 2015-05-15
AR089728A1 (en) 2014-09-10
US9334276B2 (en) 2016-05-10
EA026232B1 (en) 2017-03-31
PE23582014A1 (en) 2015-01-30
ZA201404314B (en) 2015-08-26
IN2014DN06781A (en) 2015-05-22
TW201335161A (en) 2013-09-01
EP2804863A1 (en) 2014-11-26
WO2013109514A1 (en) 2013-07-25
TWI609869B (en) 2018-01-01
RS54589B1 (en) 2016-08-31
GT201400155A (en) 2017-09-28
JP2015503627A (en) 2015-02-02
AU2013209952B2 (en) 2016-09-01
CA2863339A1 (en) 2013-07-25
SG11201404061YA (en) 2014-08-28
NZ626277A (en) 2015-10-30

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